volume 21 issue 34 pages 6903-6913

Dihydropyrrole-3-thiones: one-pot synthesis from propargylamines, acyl chlorides and sodium sulfide

Pavel A. Volkov 1
Kseniya O Khrapova 1
Ekaterina M. Vyi 1
Anton A Telezhkin 1
Ivan A Bidusenko 1
Alexander I Albanov 1
Elena Yu. Schmidt 1
Publication typeJournal Article
Publication date2023-08-09
scimago Q2
wos Q2
SJR0.600
CiteScore5.2
Impact factor2.7
ISSN14770520, 14770539
PubMed ID:  37581533
Organic Chemistry
Biochemistry
Physical and Theoretical Chemistry
Abstract
An efficient one-pot synthesis of 1,2,5-trisubstituted-1,2-dihydro-3H-pyrrole-3-thiones (up to 91% yield), representatives of essentially new heterocyclic systems, by the successive treatment of available propargylamines with acyl chlorides (PdCl2/CuI/Ph3P/Et3N, toluene, 40–45 °C, 3 h) and sodium sulfide (Na2S·9H2O, EtOH, 20–25 °C, 7 h) has been developed. The synthesis comprises the addition of sulfide anions to the formed aminoacetylenic ketones followed by dehydrative cyclization of the prototropically rearranged adducts.
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Volkov P. A. et al. Dihydropyrrole-3-thiones: one-pot synthesis from propargylamines, acyl chlorides and sodium sulfide // Organic and Biomolecular Chemistry. 2023. Vol. 21. No. 34. pp. 6903-6913.
GOST all authors (up to 50) Copy
Volkov P. A., Khrapova K. O., Vyi E. M., Telezhkin A. A., Bidusenko I. A., Albanov A. I., Schmidt E. Y., Trofimov B. A. Dihydropyrrole-3-thiones: one-pot synthesis from propargylamines, acyl chlorides and sodium sulfide // Organic and Biomolecular Chemistry. 2023. Vol. 21. No. 34. pp. 6903-6913.
RIS |
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RIS Copy
TY - JOUR
DO - 10.1039/d3ob01061a
UR - https://xlink.rsc.org/?DOI=D3OB01061A
TI - Dihydropyrrole-3-thiones: one-pot synthesis from propargylamines, acyl chlorides and sodium sulfide
T2 - Organic and Biomolecular Chemistry
AU - Volkov, Pavel A.
AU - Khrapova, Kseniya O
AU - Vyi, Ekaterina M.
AU - Telezhkin, Anton A
AU - Bidusenko, Ivan A
AU - Albanov, Alexander I
AU - Schmidt, Elena Yu.
AU - Trofimov, B. A.
PY - 2023
DA - 2023/08/09
PB - Royal Society of Chemistry (RSC)
SP - 6903-6913
IS - 34
VL - 21
PMID - 37581533
SN - 1477-0520
SN - 1477-0539
ER -
BibTex |
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BibTex (up to 50 authors) Copy
@article{2023_Volkov,
author = {Pavel A. Volkov and Kseniya O Khrapova and Ekaterina M. Vyi and Anton A Telezhkin and Ivan A Bidusenko and Alexander I Albanov and Elena Yu. Schmidt and B. A. Trofimov},
title = {Dihydropyrrole-3-thiones: one-pot synthesis from propargylamines, acyl chlorides and sodium sulfide},
journal = {Organic and Biomolecular Chemistry},
year = {2023},
volume = {21},
publisher = {Royal Society of Chemistry (RSC)},
month = {aug},
url = {https://xlink.rsc.org/?DOI=D3OB01061A},
number = {34},
pages = {6903--6913},
doi = {10.1039/d3ob01061a}
}
MLA
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MLA Copy
Volkov, Pavel A., et al. “Dihydropyrrole-3-thiones: one-pot synthesis from propargylamines, acyl chlorides and sodium sulfide.” Organic and Biomolecular Chemistry, vol. 21, no. 34, Aug. 2023, pp. 6903-6913. https://xlink.rsc.org/?DOI=D3OB01061A.
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