volume 11 issue 13 pages 3537-3545

Catalytic [4+1]-annulation of thioamides with carbenoid precursors

Publication typeJournal Article
Publication date2024-02-20
scimago Q1
wos Q1
SJR1.068
CiteScore8.2
Impact factor4.7
ISSN20524110, 20524129
Organic Chemistry
Abstract
A Rh(II)/Cu(I)-catalyzed [4 + 1]-annulation of readily available thioamides with 1-sulfonyl-1,2,3-triazoles and diazoamides was developed, delivering a general approach toward highly substituted dihydrothiophenes. A series of dihydrothiophenes having a wide diversity of functional groups, including spirocyclic, dispirocyclic and bicyclic derivatives were synthesized in high yields and good diastereoselectivity. The diastereoselectivity for the reaction of 2-(morpholino-4-carbonothioyl)-3-phenylacrylonitrile with diazoacetamides can be switched by replacing Rh(II) with a Cu(I) catalyst. Cycloalkylidene substituted thioamides formed various regioisomers under Rh(II) or Cu(I) catalysis. Furthermore, reactions of 3-diazomethylindolin-2-one with thioamides can be performed enantioselectively with ee up to 97%.
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Ilkin V. G. et al. Catalytic [4+1]-annulation of thioamides with carbenoid precursors // Organic Chemistry Frontiers. 2024. Vol. 11. No. 13. pp. 3537-3545.
GOST all authors (up to 50) Copy
Ilkin V. G., Filimonov V. O., Utepova I. A., Beryozkina T. V., Slepukhin P. A., Tumashov A. A., Dehaen W., Bakulev V. A. Catalytic [4+1]-annulation of thioamides with carbenoid precursors // Organic Chemistry Frontiers. 2024. Vol. 11. No. 13. pp. 3537-3545.
RIS |
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RIS Copy
TY - JOUR
DO - 10.1039/d3qo02025h
UR - https://xlink.rsc.org/?DOI=D3QO02025H
TI - Catalytic [4+1]-annulation of thioamides with carbenoid precursors
T2 - Organic Chemistry Frontiers
AU - Ilkin, Vladimir G
AU - Filimonov, Valeriy O
AU - Utepova, Irina A
AU - Beryozkina, Tetyana V
AU - Slepukhin, Pavel A.
AU - Tumashov, Andrey A
AU - Dehaen, Wim
AU - Bakulev, Vasiliy A.
PY - 2024
DA - 2024/02/20
PB - Royal Society of Chemistry (RSC)
SP - 3537-3545
IS - 13
VL - 11
SN - 2052-4110
SN - 2052-4129
ER -
BibTex |
Cite this
BibTex (up to 50 authors) Copy
@article{2024_Ilkin,
author = {Vladimir G Ilkin and Valeriy O Filimonov and Irina A Utepova and Tetyana V Beryozkina and Pavel A. Slepukhin and Andrey A Tumashov and Wim Dehaen and Vasiliy A. Bakulev},
title = {Catalytic [4+1]-annulation of thioamides with carbenoid precursors},
journal = {Organic Chemistry Frontiers},
year = {2024},
volume = {11},
publisher = {Royal Society of Chemistry (RSC)},
month = {feb},
url = {https://xlink.rsc.org/?DOI=D3QO02025H},
number = {13},
pages = {3537--3545},
doi = {10.1039/d3qo02025h}
}
MLA
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MLA Copy
Ilkin, Vladimir G., et al. “Catalytic [4+1]-annulation of thioamides with carbenoid precursors.” Organic Chemistry Frontiers, vol. 11, no. 13, Feb. 2024, pp. 3537-3545. https://xlink.rsc.org/?DOI=D3QO02025H.