Drug discovery: phosphinolactone, in vivo bioisostere of the lactol group
Тип публикации: Journal Article
Дата публикации: 2010-01-22
scimago Q2
wos Q2
БС1
SJR: 0.6
CiteScore: 5.2
Impact factor: 2.7
ISSN: 14770520, 14770539
PubMed ID:
20204219
Organic Chemistry
Biochemistry
Physical and Theoretical Chemistry
Краткое описание
In drug discovery, structural modifications over the lead molecule are often crucial for the development of a drug. Herein, we reported the first in vivo bioisosteric effect of phosphinolactone function in relation to the lactol group constituting the bioactive molecule: Hydroxybupropion. The preparation of phosphinolactone analogues and their antidepressant evaluation towards forced swimming test in mice showed that biological activity was regained and even strengthen.
Найдено
Ничего не найдено, попробуйте изменить настройки фильтра.
Для доступа к списку цитирований публикации необходимо авторизоваться.
Топ-30
Журналы
|
1
2
3
|
|
|
Organic Letters
3 публикации, 9.68%
|
|
|
Journal of Organic Chemistry
3 публикации, 9.68%
|
|
|
Phosphorus, Sulfur and Silicon and the Related Elements
3 публикации, 9.68%
|
|
|
Tetrahedron
2 публикации, 6.45%
|
|
|
Russian Journal of General Chemistry
2 публикации, 6.45%
|
|
|
Biomimetics
1 публикация, 3.23%
|
|
|
Molecules
1 публикация, 3.23%
|
|
|
Frontiers in Pharmacology
1 публикация, 3.23%
|
|
|
Pharmacological Research
1 публикация, 3.23%
|
|
|
Bioorganic and Medicinal Chemistry Letters
1 публикация, 3.23%
|
|
|
Mendeleev Communications
1 публикация, 3.23%
|
|
|
European Journal of Inorganic Chemistry
1 публикация, 3.23%
|
|
|
Advanced Synthesis and Catalysis
1 публикация, 3.23%
|
|
|
European Journal of Organic Chemistry
1 публикация, 3.23%
|
|
|
Journal of Medicinal Chemistry
1 публикация, 3.23%
|
|
|
Pure and Applied Chemistry
1 публикация, 3.23%
|
|
|
Topics in Current Chemistry
1 публикация, 3.23%
|
|
|
Advances in Heterocyclic Chemistry
1 публикация, 3.23%
|
|
|
Журнал Общей Химии
1 публикация, 3.23%
|
|
|
Pharmaceuticals
1 публикация, 3.23%
|
|
|
Translational Neurodegeneration
1 публикация, 3.23%
|
|
|
1
2
3
|
Издатели
|
1
2
3
4
5
6
7
|
|
|
American Chemical Society (ACS)
7 публикаций, 22.58%
|
|
|
Elsevier
5 публикаций, 16.13%
|
|
|
Wiley
4 публикации, 12.9%
|
|
|
MDPI
3 публикации, 9.68%
|
|
|
Pleiades Publishing
3 публикации, 9.68%
|
|
|
Taylor & Francis
3 публикации, 9.68%
|
|
|
Springer Nature
2 публикации, 6.45%
|
|
|
Frontiers Media S.A.
1 публикация, 3.23%
|
|
|
OOO Zhurnal "Mendeleevskie Soobshcheniya"
1 публикация, 3.23%
|
|
|
Walter de Gruyter
1 публикация, 3.23%
|
|
|
Royal Society of Chemistry (RSC)
1 публикация, 3.23%
|
|
|
1
2
3
4
5
6
7
|
- Мы не учитываем публикации, у которых нет DOI.
- Статистика публикаций обновляется еженедельно.
Вы ученый?
Создайте профиль, чтобы получать персональные рекомендации коллег, конференций и новых статей.
Метрики
31
Всего цитирований:
31
Цитирований c 2025:
5
(16.13%)
Цитировать
ГОСТ |
RIS |
BibTex |
MLA
Цитировать
ГОСТ
Скопировать
Volle J. N. et al. Drug discovery: phosphinolactone, in vivo bioisostere of the lactol group // Organic and Biomolecular Chemistry. 2010. Vol. 8. No. 6. p. 1438.
ГОСТ со всеми авторами (до 50)
Скопировать
Volle J. N., Volle J., Filippini D., Krawczy B., Kaloyanov N., van der Lee A., Maurice T., Pirat J., Virieux D. Drug discovery: phosphinolactone, in vivo bioisostere of the lactol group // Organic and Biomolecular Chemistry. 2010. Vol. 8. No. 6. p. 1438.
Цитировать
RIS
Скопировать
TY - JOUR
DO - 10.1039/b919345f
UR - https://doi.org/10.1039/b919345f
TI - Drug discovery: phosphinolactone, in vivo bioisostere of the lactol group
T2 - Organic and Biomolecular Chemistry
AU - Volle, Jean Noël
AU - Volle, Jean-Noël
AU - Filippini, Damien
AU - Krawczy, Bartlomiej
AU - Kaloyanov, Nikolay
AU - van der Lee, Arie
AU - Maurice, Tangui
AU - Pirat, Jean-Luc
AU - Virieux, David
PY - 2010
DA - 2010/01/22
PB - Royal Society of Chemistry (RSC)
SP - 1438
IS - 6
VL - 8
PMID - 20204219
SN - 1477-0520
SN - 1477-0539
ER -
Цитировать
BibTex (до 50 авторов)
Скопировать
@article{2010_Volle,
author = {Jean Noël Volle and Jean-Noël Volle and Damien Filippini and Bartlomiej Krawczy and Nikolay Kaloyanov and Arie van der Lee and Tangui Maurice and Jean-Luc Pirat and David Virieux},
title = {Drug discovery: phosphinolactone, in vivo bioisostere of the lactol group},
journal = {Organic and Biomolecular Chemistry},
year = {2010},
volume = {8},
publisher = {Royal Society of Chemistry (RSC)},
month = {jan},
url = {https://doi.org/10.1039/b919345f},
number = {6},
pages = {1438},
doi = {10.1039/b919345f}
}
Цитировать
MLA
Скопировать
Volle, Jean Noël, et al. “Drug discovery: phosphinolactone, in vivo bioisostere of the lactol group.” Organic and Biomolecular Chemistry, vol. 8, no. 6, Jan. 2010, p. 1438. https://doi.org/10.1039/b919345f.