Preparation of Novel Bridged Bicyclic Thiomorpholines as Potentially Useful Building Blocks in Medicinal Chemistry
1
Kalexsyn, Inc.
Publication type: Journal Article
Publication date: 2013-09-12
scimago Q2
wos Q2
SJR: 0.559
CiteScore: 4.6
Impact factor: 2.3
ISSN: 00397881, 1437210X
Catalysis
Organic Chemistry
Abstract
Thiomorpholine and thiomorpholine 1,1-dioxide are important building blocks in medicinal chemistry research, and some analogues containing these moieties have entered human clinical trials. Analogues containing bridged bicyclic thiomorpholines have also shown interesting biological profiles. 3-Thia-6-azabicyclo[3.1.1]heptane, 3-thia-8-azabicyclo[3.2.1]octane, and their corresponding 1,1-dioxide counterparts were prepared as novel bicyclic thiomorpholine building blocks. Each heterocycle was synthesized from an inexpensive starting material by straightforward chemistry.
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Walker D., Rogier D. Preparation of Novel Bridged Bicyclic Thiomorpholines as Potentially Useful Building Blocks in Medicinal Chemistry // Synthesis. 2013. Vol. 45. No. 21. pp. 2966-2970.
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Walker D., Rogier D. Preparation of Novel Bridged Bicyclic Thiomorpholines as Potentially Useful Building Blocks in Medicinal Chemistry // Synthesis. 2013. Vol. 45. No. 21. pp. 2966-2970.
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RIS
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TY - JOUR
DO - 10.1055/s-0033-1338528
UR - https://doi.org/10.1055/s-0033-1338528
TI - Preparation of Novel Bridged Bicyclic Thiomorpholines as Potentially Useful Building Blocks in Medicinal Chemistry
T2 - Synthesis
AU - Walker, Daniel
AU - Rogier, D
PY - 2013
DA - 2013/09/12
PB - Georg Thieme Verlag KG
SP - 2966-2970
IS - 21
VL - 45
SN - 0039-7881
SN - 1437-210X
ER -
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BibTex (up to 50 authors)
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@article{2013_Walker,
author = {Daniel Walker and D Rogier},
title = {Preparation of Novel Bridged Bicyclic Thiomorpholines as Potentially Useful Building Blocks in Medicinal Chemistry},
journal = {Synthesis},
year = {2013},
volume = {45},
publisher = {Georg Thieme Verlag KG},
month = {sep},
url = {https://doi.org/10.1055/s-0033-1338528},
number = {21},
pages = {2966--2970},
doi = {10.1055/s-0033-1338528}
}
Cite this
MLA
Copy
Walker, Daniel, and D Rogier. “Preparation of Novel Bridged Bicyclic Thiomorpholines as Potentially Useful Building Blocks in Medicinal Chemistry.” Synthesis, vol. 45, no. 21, Sep. 2013, pp. 2966-2970. https://doi.org/10.1055/s-0033-1338528.