issue 24 pages 4175-4182

Novel macrocyclic bile acid derivatives; Selective and easy binding of two cholic acid moieties at the 3-and 3'-positions

Nikolay Lukashev
Alexey Kazantsev
Pavel Donez
Mikhail Baranov
Elina Sievänen
Erkki Kolehmainen
Publication typeJournal Article
Publication date2009-10-19
scimago Q2
wos Q2
SJR0.559
CiteScore4.6
Impact factor2.3
ISSN00397881, 1437210X
Catalysis
Organic Chemistry
Abstract
The synthesis of macrocyclic derivatives of bile acids (cholaphanes) is elaborated using the formation of ester or amide linkages at the 3α,3'α- and 24,24'-positions of lithocholic, deoxycholic or cholic acids. The conditions were found under which the selective diacylation at the 3α,3'α- and 24,24'-positions of two molecules of cholic acid by dichloroanhydrides of arene(hetarene)dicarboxylic acid proceeds in good yields without prior protection of the 7α- and 12α-hydroxy groups.
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Lukashev N. et al. Novel macrocyclic bile acid derivatives; Selective and easy binding of two cholic acid moieties at the 3-and 3'-positions // Synthesis. 2009. Vol. 24. pp. 4175-4182.
GOST all authors (up to 50) Copy
Lukashev N., Kazantsev A., Averin A., Donez P., Baranov M., Sievänen E., Kolehmainen E., Averin A. A. Novel macrocyclic bile acid derivatives; Selective and easy binding of two cholic acid moieties at the 3-and 3'-positions // Synthesis. 2009. Vol. 24. pp. 4175-4182.
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RIS Copy
TY - JOUR
DO - 10.1055/s-0029-1217057
UR - https://doi.org/10.1055/s-0029-1217057
TI - Novel macrocyclic bile acid derivatives; Selective and easy binding of two cholic acid moieties at the 3-and 3'-positions
T2 - Synthesis
AU - Lukashev, Nikolay
AU - Kazantsev, Alexey
AU - Averin, Alexey
AU - Donez, Pavel
AU - Baranov, Mikhail
AU - Sievänen, Elina
AU - Kolehmainen, Erkki
AU - Averin, Alexey A
PY - 2009
DA - 2009/10/19
PB - Georg Thieme Verlag KG
SP - 4175-4182
IS - 24
SN - 0039-7881
SN - 1437-210X
ER -
BibTex
Cite this
BibTex (up to 50 authors) Copy
@article{2009_Lukashev,
author = {Nikolay Lukashev and Alexey Kazantsev and Alexey Averin and Pavel Donez and Mikhail Baranov and Elina Sievänen and Erkki Kolehmainen and Alexey A Averin},
title = {Novel macrocyclic bile acid derivatives; Selective and easy binding of two cholic acid moieties at the 3-and 3'-positions},
journal = {Synthesis},
year = {2009},
publisher = {Georg Thieme Verlag KG},
month = {oct},
url = {https://doi.org/10.1055/s-0029-1217057},
number = {24},
pages = {4175--4182},
doi = {10.1055/s-0029-1217057}
}
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