SYNTHESIS, ANTI-BACTERIAL AND ANTIOXIDANT PROPERTIES OF ETHYL 7-AMINO-3-BENZOYL-2-METHYLINDOLIZINE-1-CARBOXYLATE DERIVATIVES.

Тип публикацииProceedings Article
Дата публикации2020-10-06
SJR0.146
CiteScore0.7
Impact factor
ISSN0094243X, 15517616
Краткое описание
An efficient synthesis of novel ethyl 7-amino-3-benzoylindolizine-1-carboxylate derivatives has been described using 4-aminopyridine and different phenacyl bromides in acetone and fallowed by reacting with electron-deficient acetylenes in the presence of potassium carbonate base with anhydrous DMF solvent. The structures of newly synthesized compounds have been confirmed by spectroscopic techniques and studied there in vitro antioxidant properties using a DPPH scavenging method. The compound ethyl 7-amino-3-(4-methoxybenzoyl) indolizine-1-carboxylate has shown good antioxidant potent. The compound ethyl 7-amino-3-(4-methoxybenzoyl)indolizine-1-carboxylate, ethyl 7-amino-3-(4-bromobenzoyl)indolizine-1-carboxylate and ethyl 7-amino-3-(4-chlorobenzoyl)indolizine-1-carboxylate has very potent to anti-bacterial activity.
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Journal of Molecular Structure
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Uppar V. et al. SYNTHESIS, ANTI-BACTERIAL AND ANTIOXIDANT PROPERTIES OF ETHYL 7-AMINO-3-BENZOYL-2-METHYLINDOLIZINE-1-CARBOXYLATE DERIVATIVES. // AIP Conference Proceedings. 2020.
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Uppar V., Basarikatti A. I., Padmashali B., Chandrashekharappa S., Chougala M., Mudnakudu Nagaraju K. K., Mohan M. K., Banuprakash G., Ningegowda R., Rachotimath B. B. SYNTHESIS, ANTI-BACTERIAL AND ANTIOXIDANT PROPERTIES OF ETHYL 7-AMINO-3-BENZOYL-2-METHYLINDOLIZINE-1-CARBOXYLATE DERIVATIVES. // AIP Conference Proceedings. 2020.
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TY - CPAPER
DO - 10.1063/5.0022905
UR - https://doi.org/10.1063/5.0022905
TI - SYNTHESIS, ANTI-BACTERIAL AND ANTIOXIDANT PROPERTIES OF ETHYL 7-AMINO-3-BENZOYL-2-METHYLINDOLIZINE-1-CARBOXYLATE DERIVATIVES.
T2 - AIP Conference Proceedings
AU - Uppar, Vijayakumar
AU - Basarikatti, Atiyaparveen I
AU - Padmashali, Basavaraj
AU - Chandrashekharappa, Sandeep
AU - Chougala, Mallikarjun
AU - Mudnakudu Nagaraju, Kiran K
AU - Mohan, Mahendra K.
AU - Banuprakash, Govindappa
AU - Ningegowda, Raghu
AU - Rachotimath, Beena B
PY - 2020
DA - 2020/10/06
PB - AIP Publishing
SN - 0094-243X
SN - 1551-7616
ER -
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@inproceedings{2020_Uppar,
author = {Vijayakumar Uppar and Atiyaparveen I Basarikatti and Basavaraj Padmashali and Sandeep Chandrashekharappa and Mallikarjun Chougala and Kiran K Mudnakudu Nagaraju and Mahendra K. Mohan and Govindappa Banuprakash and Raghu Ningegowda and Beena B Rachotimath},
title = {SYNTHESIS, ANTI-BACTERIAL AND ANTIOXIDANT PROPERTIES OF ETHYL 7-AMINO-3-BENZOYL-2-METHYLINDOLIZINE-1-CARBOXYLATE DERIVATIVES.},
year = {2020},
month = {oct},
publisher = {AIP Publishing}
}
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