Open Access
Azoloazines as A2a receptor antagonists. Structure–activity relationship
Тип публикации: Journal Article
Дата публикации: 2018-07-01
SCImago Q1
WOS Q1
БС1
SJR: 0.955
CiteScore: 10.5
Impact factor: 7.1
ISSN: 0036021X, 14684837
General Chemistry
Краткое описание
Non-xanthine inhibitors of the adenosine A2a receptor of the azoloazine series are good candidates for use as drugs for the treatment of neurodegenerative diseases and sepsis. This review systematizes and summarizes the structure – activity relationships in the series of triazoloazines, including annulated pyrimidines, pyrazines and triazines, as well as their tricyclic fused analogues. The above relationships for such systems are analyzed. The structures of the most efficient functional moieties from the point of view of affinity for the A2a receptor and selectivity for other types of adenosine receptors (A1, A2b, A3) are presented.
The bibliography includes 71 references.
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Savateev K. V. et al. Azoloazines as A2a receptor antagonists. Structure–activity relationship // Russian Chemical Reviews. 2018. Vol. 87. No. 7. pp. 636-669.
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Savateev K. V., Ulomsky E. N., Butorin I. I., Charushin V. N., Rusinov V. L., Chupakhin O. N. Azoloazines as A2a receptor antagonists. Structure–activity relationship // Russian Chemical Reviews. 2018. Vol. 87. No. 7. pp. 636-669.
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TY - JOUR
DO - 10.1070/RCR4792
UR - https://doi.org/10.1070/RCR4792
TI - Azoloazines as A2a receptor antagonists. Structure–activity relationship
T2 - Russian Chemical Reviews
AU - Savateev, Konstantin V
AU - Ulomsky, Evgeny N
AU - Butorin, Ilya I
AU - Charushin, Valery N.
AU - Rusinov, Vladimir L.
AU - Chupakhin, Oleg N.
PY - 2018
DA - 2018/07/01
PB - Autonomous Non-profit Organization Editorial Board of the journal Uspekhi Khimii
SP - 636-669
IS - 7
VL - 87
SN - 0036-021X
SN - 1468-4837
ER -
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@article{2018_Savateev,
author = {Konstantin V Savateev and Evgeny N Ulomsky and Ilya I Butorin and Valery N. Charushin and Vladimir L. Rusinov and Oleg N. Chupakhin},
title = {Azoloazines as A2a receptor antagonists. Structure–activity relationship},
journal = {Russian Chemical Reviews},
year = {2018},
volume = {87},
publisher = {Autonomous Non-profit Organization Editorial Board of the journal Uspekhi Khimii},
month = {jul},
url = {https://doi.org/10.1070/RCR4792},
number = {7},
pages = {636--669},
doi = {10.1070/RCR4792}
}
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MLA
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Savateev, Konstantin V., et al. “Azoloazines as A2a receptor antagonists. Structure–activity relationship.” Russian Chemical Reviews, vol. 87, no. 7, Jul. 2018, pp. 636-669. https://doi.org/10.1070/RCR4792.
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