Anticonvulsant Activity and Toxicity of Phensuximide, Methsuximide and Ethosuximide
1
Research Division, Parke, Davis and Company, Ann Arbor, Mich. (U.S.A.)
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Тип публикации: Journal Article
Дата публикации: 1963-12-01
scimago Q1
wos Q1
БС1
SJR: 2.371
CiteScore: 11.4
Impact factor: 6.6
ISSN: 00139580, 15281167, 15281157
PubMed ID:
14020499
Neurology
Neurology (clinical)
Краткое описание
The anticonvulsant properties and toxicity of phensuximide (Milontin), methsuximide (Celontin) and ethosuximide (Zarontin) have been investigated in laboratory animals. The three compounds were very effective in suppressing the initial clonic seizures induced by Metrazol in rats and mice. Whereas methsuximide and phensuximide were capable of protecting mice from tonic extensor seizures to supramaximal electroshock at non‐neurotoxic and slightly ataxic doses respectively, ethosuximide could do so only at anesthetic dose levels. The anticonvulsant spectrum of methsuximide was shown to be similar to that of phenacemide; ethosuximide, on the other hand, resembles trimethadione very closely in anticonvulsant action. A discussion was given to correlate the anticonvulsant properties of these drugs as examined in mice and their therapeutic indications for the management of petit mal, grand mal and psychomotor epilepsy.
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Chen G., Weston J. K., Bratton A. Anticonvulsant Activity and Toxicity of Phensuximide, Methsuximide and Ethosuximide // Epilepsia. 1963. Vol. 4. No. 1-4. pp. 66-76.
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Chen G., Weston J. K., Bratton A. Anticonvulsant Activity and Toxicity of Phensuximide, Methsuximide and Ethosuximide // Epilepsia. 1963. Vol. 4. No. 1-4. pp. 66-76.
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TY - JOUR
DO - 10.1111/j.1528-1157.1963.tb05209.x
UR - https://doi.org/10.1111/j.1528-1157.1963.tb05209.x
TI - Anticonvulsant Activity and Toxicity of Phensuximide, Methsuximide and Ethosuximide
T2 - Epilepsia
AU - Chen, G.
AU - Weston, J K
AU - Bratton, A.C.
PY - 1963
DA - 1963/12/01
PB - Wiley
SP - 66-76
IS - 1-4
VL - 4
PMID - 14020499
SN - 0013-9580
SN - 1528-1167
SN - 1528-1157
ER -
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@article{1963_Chen,
author = {G. Chen and J K Weston and A.C. Bratton},
title = {Anticonvulsant Activity and Toxicity of Phensuximide, Methsuximide and Ethosuximide},
journal = {Epilepsia},
year = {1963},
volume = {4},
publisher = {Wiley},
month = {dec},
url = {https://doi.org/10.1111/j.1528-1157.1963.tb05209.x},
number = {1-4},
pages = {66--76},
doi = {10.1111/j.1528-1157.1963.tb05209.x}
}
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MLA
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Chen, G., et al. “Anticonvulsant Activity and Toxicity of Phensuximide, Methsuximide and Ethosuximide.” Epilepsia, vol. 4, no. 1-4, Dec. 1963, pp. 66-76. https://doi.org/10.1111/j.1528-1157.1963.tb05209.x.