Antifungal Agents. Part 3: Synthesis and Antifungal Activities of 3-Acylindole Analogs against Phytopathogenic Fungi In Vitro
Publication type: Journal Article
Publication date: 2011-09-15
scimago Q2
wos Q2
SJR: 0.689
CiteScore: 5.6
Impact factor: 3.3
ISSN: 17470277, 17470285
PubMed ID:
21827634
Organic Chemistry
Drug Discovery
Biochemistry
Pharmacology
Molecular Medicine
Abstract
To find more potent antifungal compounds, twenty 3-acylindole analogs were synthesized and bio-evaluated for their antifungal activities against seven phytopathogenic fungi. Structure-activity relationships investigations revealed that 4- or 6-methyl and 3-acetyl or propionyl groups were the important structural properties of 3-acylindoles for the activities. Especially 4-methyl-3-propionylindole, 12, displayed the more potent activities than hymexazol, a commercially available agricultural fungicide, and might be considered as a new promising lead candidate for further design and synthesis of agricultural fungicides.
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GOST
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Xu H., Bin Yang W., Wang Q. Antifungal Agents. Part 3: Synthesis and Antifungal Activities of 3-Acylindole Analogs against Phytopathogenic Fungi In Vitro // Chemical Biology and Drug Design. 2011. Vol. 78. No. 5. pp. 864-868.
GOST all authors (up to 50)
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Xu H., Bin Yang W., Wang Q. Antifungal Agents. Part 3: Synthesis and Antifungal Activities of 3-Acylindole Analogs against Phytopathogenic Fungi In Vitro // Chemical Biology and Drug Design. 2011. Vol. 78. No. 5. pp. 864-868.
Cite this
RIS
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TY - JOUR
DO - 10.1111/j.1747-0285.2011.01212.x
UR - https://doi.org/10.1111/j.1747-0285.2011.01212.x
TI - Antifungal Agents. Part 3: Synthesis and Antifungal Activities of 3-Acylindole Analogs against Phytopathogenic Fungi In Vitro
T2 - Chemical Biology and Drug Design
AU - Xu, Hui
AU - Bin Yang, Wen
AU - Wang, Qin
PY - 2011
DA - 2011/09/15
PB - Wiley
SP - 864-868
IS - 5
VL - 78
PMID - 21827634
SN - 1747-0277
SN - 1747-0285
ER -
Cite this
BibTex (up to 50 authors)
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@article{2011_Xu,
author = {Hui Xu and Wen Bin Yang and Qin Wang},
title = {Antifungal Agents. Part 3: Synthesis and Antifungal Activities of 3-Acylindole Analogs against Phytopathogenic Fungi In Vitro},
journal = {Chemical Biology and Drug Design},
year = {2011},
volume = {78},
publisher = {Wiley},
month = {sep},
url = {https://doi.org/10.1111/j.1747-0285.2011.01212.x},
number = {5},
pages = {864--868},
doi = {10.1111/j.1747-0285.2011.01212.x}
}
Cite this
MLA
Copy
Xu, Hui, et al. “Antifungal Agents. Part 3: Synthesis and Antifungal Activities of 3-Acylindole Analogs against Phytopathogenic Fungi In Vitro.” Chemical Biology and Drug Design, vol. 78, no. 5, Sep. 2011, pp. 864-868. https://doi.org/10.1111/j.1747-0285.2011.01212.x.