volume 90 issue 9 pages 1581-1590

Synthesis and Analgesic Activity of N,6-Diaryl-4-hydroxy-4-methyl-2-oxocyclohexane-1-carboxamides and Their Dehydration Products

Publication typeJournal Article
Publication date2020-09-01
scimago Q4
wos Q4
SJR0.179
CiteScore1.4
Impact factor0.8
ISSN10703632, 16083350
General Chemistry
Abstract
A series of new N,6-diaryl-4-hydroxy-4-methyl-2-oxocyclohexane-1-carboxamides was obtained through the reaction of N-arylamides of acetoacetic acid with benzalacetone and 4-chlorobenzalacetone under basic conditions (KOH) in methanol at room temperature. Increasing of the amount of potassium hydroxide used in the reaction led to the formation of dehydration products, namely N,6-diaryl-4-methyl-2-oxocyclohex-3-ene-1-carboxamides. The latter were also formed by using unsubstituted acetoacetamide and N-methylacetoacetamide. The synthesized compounds were tested for analgesic activity.
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Nosova N. V. et al. Synthesis and Analgesic Activity of N,6-Diaryl-4-hydroxy-4-methyl-2-oxocyclohexane-1-carboxamides and Their Dehydration Products // Russian Journal of General Chemistry. 2020. Vol. 90. No. 9. pp. 1581-1590.
GOST all authors (up to 50) Copy
Nosova N. V., Sokolov A. A., Gein O. N., Gein V. L., Yankin A. N., Danilov S. E., Dmitriev M. V. Synthesis and Analgesic Activity of N,6-Diaryl-4-hydroxy-4-methyl-2-oxocyclohexane-1-carboxamides and Their Dehydration Products // Russian Journal of General Chemistry. 2020. Vol. 90. No. 9. pp. 1581-1590.
RIS |
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RIS Copy
TY - JOUR
DO - 10.1134/S1070363220090017
UR - https://doi.org/10.1134/S1070363220090017
TI - Synthesis and Analgesic Activity of N,6-Diaryl-4-hydroxy-4-methyl-2-oxocyclohexane-1-carboxamides and Their Dehydration Products
T2 - Russian Journal of General Chemistry
AU - Nosova, N V
AU - Sokolov, A. A.
AU - Gein, O N
AU - Gein, V L
AU - Yankin, A N
AU - Danilov, S E
AU - Dmitriev, M V
PY - 2020
DA - 2020/09/01
PB - Pleiades Publishing
SP - 1581-1590
IS - 9
VL - 90
SN - 1070-3632
SN - 1608-3350
ER -
BibTex |
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BibTex (up to 50 authors) Copy
@article{2020_Nosova,
author = {N V Nosova and A. A. Sokolov and O N Gein and V L Gein and A N Yankin and S E Danilov and M V Dmitriev},
title = {Synthesis and Analgesic Activity of N,6-Diaryl-4-hydroxy-4-methyl-2-oxocyclohexane-1-carboxamides and Their Dehydration Products},
journal = {Russian Journal of General Chemistry},
year = {2020},
volume = {90},
publisher = {Pleiades Publishing},
month = {sep},
url = {https://doi.org/10.1134/S1070363220090017},
number = {9},
pages = {1581--1590},
doi = {10.1134/S1070363220090017}
}
MLA
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MLA Copy
Nosova, N. V., et al. “Synthesis and Analgesic Activity of N,6-Diaryl-4-hydroxy-4-methyl-2-oxocyclohexane-1-carboxamides and Their Dehydration Products.” Russian Journal of General Chemistry, vol. 90, no. 9, Sep. 2020, pp. 1581-1590. https://doi.org/10.1134/S1070363220090017.