volume 71 issue 9 pages 1021-1026

Hepatitis C virus RNA-dependent RNA polymerase: Study on the inhibition mechanism by pyrogallol derivatives

M. V. Kozlov 1
K. M. Polyakov 1
Ivanov A.V. 1
S E Filippova 1
A O Kuzyakin 1
V L Tunitskaya 1
Publication typeJournal Article
Publication date2006-09-21
scimago Q2
wos Q4
SJR0.659
CiteScore3.8
Impact factor2.2
ISSN00062979, 16083040
Biochemistry
General Medicine
Abstract
Pyrogallol reversibly and noncompetitively inhibits the activity of the hepatitis C RNA-dependent RNA polyme rase. Based on molecular modeling of the inhibitor binding in the active site of the enzyme, the inhibition was suggested to be realized via chelation of two magnesium cations involved in the catalysis at the stage of the phosphoryl residue transfer. The proposed model allowed us to purposefully synthesize new derivatives with higher inhibitory capacity.
Found 
Found 

Top-30

Journals

1
Biochemistry (Moscow)
1 publication, 25%
Sensors
1 publication, 25%
Biochimie
1 publication, 25%
Handbook of Experimental Pharmacology
1 publication, 25%
1

Publishers

1
Pleiades Publishing
1 publication, 25%
MDPI
1 publication, 25%
Elsevier
1 publication, 25%
Springer Nature
1 publication, 25%
1
  • We do not take into account publications without a DOI.
  • Statistics recalculated weekly.

Are you a researcher?

Create a profile to get free access to personal recommendations for colleagues and new articles.
Metrics
4
Share
Cite this
GOST |
Cite this
GOST Copy
Kozlov M. V. et al. Hepatitis C virus RNA-dependent RNA polymerase: Study on the inhibition mechanism by pyrogallol derivatives // Biochemistry (Moscow). 2006. Vol. 71. No. 9. pp. 1021-1026.
GOST all authors (up to 50) Copy
Kozlov M. V., Polyakov K. M., A.V. I., Filippova S. E., Kuzyakin A. O., Tunitskaya V. L., Kochetkov S. N. Hepatitis C virus RNA-dependent RNA polymerase: Study on the inhibition mechanism by pyrogallol derivatives // Biochemistry (Moscow). 2006. Vol. 71. No. 9. pp. 1021-1026.
RIS |
Cite this
RIS Copy
TY - JOUR
DO - 10.1134/S0006297906090112
UR - https://doi.org/10.1134/S0006297906090112
TI - Hepatitis C virus RNA-dependent RNA polymerase: Study on the inhibition mechanism by pyrogallol derivatives
T2 - Biochemistry (Moscow)
AU - Kozlov, M. V.
AU - Polyakov, K. M.
AU - A.V., Ivanov
AU - Filippova, S E
AU - Kuzyakin, A O
AU - Tunitskaya, V L
AU - Kochetkov, S. N.
PY - 2006
DA - 2006/09/21
PB - Pleiades Publishing
SP - 1021-1026
IS - 9
VL - 71
PMID - 17009957
SN - 0006-2979
SN - 1608-3040
ER -
BibTex |
Cite this
BibTex (up to 50 authors) Copy
@article{2006_Kozlov,
author = {M. V. Kozlov and K. M. Polyakov and Ivanov A.V. and S E Filippova and A O Kuzyakin and V L Tunitskaya and S. N. Kochetkov},
title = {Hepatitis C virus RNA-dependent RNA polymerase: Study on the inhibition mechanism by pyrogallol derivatives},
journal = {Biochemistry (Moscow)},
year = {2006},
volume = {71},
publisher = {Pleiades Publishing},
month = {sep},
url = {https://doi.org/10.1134/S0006297906090112},
number = {9},
pages = {1021--1026},
doi = {10.1134/S0006297906090112}
}
MLA
Cite this
MLA Copy
Kozlov, M. V., et al. “Hepatitis C virus RNA-dependent RNA polymerase: Study on the inhibition mechanism by pyrogallol derivatives.” Biochemistry (Moscow), vol. 71, no. 9, Sep. 2006, pp. 1021-1026. https://doi.org/10.1134/S0006297906090112.