том 42 издание 2 страницы 191-197

Synthesis of (Z)-N-hydroxy-3-methoxy-3-phenylacrylamide as new selective inhibitor of hepatitis C virus replication

Тип публикацииJournal Article
Дата публикации2016-03-01
scimago Q4
wos Q3
white level БС2
SJR0.267
CiteScore1.9
Impact factor1.7
ISSN10681620, 1608330X, 15739163
Organic Chemistry
Biochemistry
Краткое описание
According to recently published results, cinnamic hydroxamic acid (CHA) inhibits replication of hepatitis C virus (HCV). We synthesized a structural analogue of CHA, i.e., (Z)-N-hydroxy-3-methoxy3-phenylacrylamide, which inhibited HCV replication five times more selectively than CHA. It was found that both compounds did not inhibit deacetylation of Ac-α-tubulin with histone deacetylase 6, the activity of which is important for virus replication.
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European Journal of Medicinal Chemistry
1 публикация, 33.33%
Russian Journal of Bioorganic Chemistry
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Current Organic Chemistry
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Elsevier
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Pleiades Publishing
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Bentham Science Publishers Ltd.
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ГОСТ |
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Kozlov M. V. et al. Synthesis of (Z)-N-hydroxy-3-methoxy-3-phenylacrylamide as new selective inhibitor of hepatitis C virus replication // Russian Journal of Bioorganic Chemistry. 2016. Vol. 42. No. 2. pp. 191-197.
ГОСТ со всеми авторами (до 50) Скопировать
Kozlov M. V., Kleymenova A. A., Konduktorov K. A., Malikova A. Z., Kamarova K. A., Novikov R. A., Kochetkov S. N. Synthesis of (Z)-N-hydroxy-3-methoxy-3-phenylacrylamide as new selective inhibitor of hepatitis C virus replication // Russian Journal of Bioorganic Chemistry. 2016. Vol. 42. No. 2. pp. 191-197.
RIS |
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TY - JOUR
DO - 10.1134/S1068162016010076
UR - https://doi.org/10.1134/S1068162016010076
TI - Synthesis of (Z)-N-hydroxy-3-methoxy-3-phenylacrylamide as new selective inhibitor of hepatitis C virus replication
T2 - Russian Journal of Bioorganic Chemistry
AU - Kozlov, M. V.
AU - Kleymenova, A A
AU - Konduktorov, K A
AU - Malikova, A Z
AU - Kamarova, K A
AU - Novikov, R A
AU - Kochetkov, S. N.
PY - 2016
DA - 2016/03/01
PB - Pleiades Publishing
SP - 191-197
IS - 2
VL - 42
SN - 1068-1620
SN - 1608-330X
SN - 1573-9163
ER -
BibTex |
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@article{2016_Kozlov,
author = {M. V. Kozlov and A A Kleymenova and K A Konduktorov and A Z Malikova and K A Kamarova and R A Novikov and S. N. Kochetkov},
title = {Synthesis of (Z)-N-hydroxy-3-methoxy-3-phenylacrylamide as new selective inhibitor of hepatitis C virus replication},
journal = {Russian Journal of Bioorganic Chemistry},
year = {2016},
volume = {42},
publisher = {Pleiades Publishing},
month = {mar},
url = {https://doi.org/10.1134/S1068162016010076},
number = {2},
pages = {191--197},
doi = {10.1134/S1068162016010076}
}
MLA
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Kozlov, M. V., et al. “Synthesis of (Z)-N-hydroxy-3-methoxy-3-phenylacrylamide as new selective inhibitor of hepatitis C virus replication.” Russian Journal of Bioorganic Chemistry, vol. 42, no. 2, Mar. 2016, pp. 191-197. https://doi.org/10.1134/S1068162016010076.
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