Open Access
Natural Product Communications, volume 14, issue 7, pages 1934578X1986067
Synthesis and сytotoxicity of a-azepanobetulinic acid N-methyl-piperazinylamide
Giniyatullina Gulnara V
1
,
Kazakova Oxana B.
1
,
Baikova Irina P
1
,
Yamansarov Emil Yu
2
,
Osterman Ilya A.
2, 3, 4
,
Komarova Ekaterina S.
2, 3
,
Saltikova Irina V
2
,
Majouga Alexander G.
2, 5, 6
,
Ivanenkov Yan A
7, 8
7
Publication type: Journal Article
Publication date: 2019-07-30
Journal:
Natural Product Communications
Quartile SCImago
Q3
Quartile WOS
Q4
Impact factor: 1.8
ISSN: 1934578X, 15559475
Drug Discovery
General Medicine
Pharmacology
Complementary and alternative medicine
Plant Science
Abstract
The synthesis of A-azepanobetulinic acid N-methylpiperazinylamide was performed through a series of transformations (oximation, Beckmann rearrangement, reduction) of previously synthesized betulonic acid N-methylpiperazinylamide. In vitro cytotoxic activity was detected for the obtained compound against a number of cancer cell lines, and its potential was revealed as an antibacterial agent.
Citations by journals
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1
2
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International Journal of Molecular Sciences
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International Journal of Molecular Sciences
2 publications, 40%
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Molecules
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Molecules
1 publication, 20%
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Medicinal Chemistry Research
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Medicinal Chemistry Research
1 publication, 20%
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Russian Journal of Organic Chemistry
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Russian Journal of Organic Chemistry
1 publication, 20%
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1
2
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Citations by publishers
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1
2
3
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Multidisciplinary Digital Publishing Institute (MDPI)
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Multidisciplinary Digital Publishing Institute (MDPI)
3 publications, 60%
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Springer Nature
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Springer Nature
1 publication, 20%
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Pleiades Publishing
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Pleiades Publishing
1 publication, 20%
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1
2
3
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- We do not take into account publications that without a DOI.
- Statistics recalculated only for publications connected to researchers, organizations and labs registered on the platform.
- Statistics recalculated weekly.
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Giniyatullina G. V. et al. Synthesis and сytotoxicity of a-azepanobetulinic acid N-methyl-piperazinylamide // Natural Product Communications. 2019. Vol. 14. No. 7. p. 1934578X1986067.
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Giniyatullina G. V., Kazakova O. B., Baikova I. P., Yamansarov E. Yu., Osterman I. A., Komarova E. S., Skvortsov D. A., Saltikova I. V., Majouga A. G., Ivanenkov Y. A. Synthesis and сytotoxicity of a-azepanobetulinic acid N-methyl-piperazinylamide // Natural Product Communications. 2019. Vol. 14. No. 7. p. 1934578X1986067.
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TY - JOUR
DO - 10.1177/1934578X19860670
UR - https://doi.org/10.1177%2F1934578X19860670
TI - Synthesis and сytotoxicity of a-azepanobetulinic acid N-methyl-piperazinylamide
T2 - Natural Product Communications
AU - Giniyatullina, Gulnara V
AU - Baikova, Irina P
AU - Osterman, Ilya A.
AU - Komarova, Ekaterina S.
AU - Skvortsov, Dmitry A.
AU - Saltikova, Irina V
AU - Majouga, Alexander G.
AU - Kazakova, Oxana B.
AU - Yamansarov, Emil Yu
AU - Ivanenkov, Yan A
PY - 2019
DA - 2019/07/30 00:00:00
PB - SAGE
SP - 1934578X1986067
IS - 7
VL - 14
SN - 1934-578X
SN - 1555-9475
ER -
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@article{2019_Giniyatullina,
author = {Gulnara V Giniyatullina and Irina P Baikova and Ilya A. Osterman and Ekaterina S. Komarova and Dmitry A. Skvortsov and Irina V Saltikova and Alexander G. Majouga and Oxana B. Kazakova and Emil Yu Yamansarov and Yan A Ivanenkov},
title = {Synthesis and сytotoxicity of a-azepanobetulinic acid N-methyl-piperazinylamide},
journal = {Natural Product Communications},
year = {2019},
volume = {14},
publisher = {SAGE},
month = {jul},
url = {https://doi.org/10.1177%2F1934578X19860670},
number = {7},
pages = {1934578X1986067},
doi = {10.1177/1934578X19860670}
}
Cite this
MLA
Copy
Giniyatullina, Gulnara V., et al. “Synthesis and сytotoxicity of a-azepanobetulinic acid N-methyl-piperazinylamide.” Natural Product Communications, vol. 14, no. 7, Jul. 2019, p. 1934578X1986067. https://doi.org/10.1177%2F1934578X19860670.