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Recent Progress in the Development of Synthetic Hybrids of Natural or Unnatural Bioactive Compounds for Medicinal Chemistry

Тип публикацииJournal Article
Дата публикации2010-06-27
scimago Q2
wos Q3
БС1
SJR0.662
CiteScore8.5
Impact factor3.3
ISSN13895575, 18755607
Drug Discovery
General Medicine
Pharmacology
Краткое описание
The present mini-review highlights the recent developments on different classes of synthetic hybrids of natural and/or unnatural bioactive compounds, the utilization of which is very promising, as distinct features of each component can be hybridized and their properties leveraged. Particular stress is put on the respective mode of action and the corresponding rationale behind covalent combinations of various bioactive agents to increase their therapeutic potential, facilitate their administration, to reduce harmful side effects and/or to overcome the problem of multi-drug resistance. This rather recent approach has already found applications in the development of new anti-cancer, anti-Alzheimer, anti-malaria, anti-microbial therapeutics and other novel compounds with unprecedented bioactivity.
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ГОСТ |
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Tsogoeva S. B. Recent Progress in the Development of Synthetic Hybrids of Natural or Unnatural Bioactive Compounds for Medicinal Chemistry // Mini-Reviews in Medicinal Chemistry. 2010. Vol. 10. No. 9. pp. 773-793.
ГОСТ со всеми авторами (до 50) Скопировать
Tsogoeva S. B. Recent Progress in the Development of Synthetic Hybrids of Natural or Unnatural Bioactive Compounds for Medicinal Chemistry // Mini-Reviews in Medicinal Chemistry. 2010. Vol. 10. No. 9. pp. 773-793.
RIS |
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TY - JOUR
DO - 10.2174/138955710791608280
UR - https://doi.org/10.2174/138955710791608280
TI - Recent Progress in the Development of Synthetic Hybrids of Natural or Unnatural Bioactive Compounds for Medicinal Chemistry
T2 - Mini-Reviews in Medicinal Chemistry
AU - Tsogoeva, Svetlana B.
PY - 2010
DA - 2010/06/27
PB - Bentham Science Publishers Ltd.
SP - 773-793
IS - 9
VL - 10
PMID - 20105118
SN - 1389-5575
SN - 1875-5607
ER -
BibTex |
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BibTex (до 50 авторов) Скопировать
@article{2010_Tsogoeva,
author = {Svetlana B. Tsogoeva},
title = {Recent Progress in the Development of Synthetic Hybrids of Natural or Unnatural Bioactive Compounds for Medicinal Chemistry},
journal = {Mini-Reviews in Medicinal Chemistry},
year = {2010},
volume = {10},
publisher = {Bentham Science Publishers Ltd.},
month = {jun},
url = {https://doi.org/10.2174/138955710791608280},
number = {9},
pages = {773--793},
doi = {10.2174/138955710791608280}
}
MLA
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Tsogoeva, Svetlana B.. “Recent Progress in the Development of Synthetic Hybrids of Natural or Unnatural Bioactive Compounds for Medicinal Chemistry.” Mini-Reviews in Medicinal Chemistry, vol. 10, no. 9, Jun. 2010, pp. 773-793. https://doi.org/10.2174/138955710791608280.