том 75 издание 4 страницы 218-224

Physical and Chemical Properties of the Guest–Host Inclusion Complexes of Cyprofloxacin with β-Cyclodextrin Derivatives

Тип публикацииJournal Article
Дата публикации2020-07-01
scimago Q4
wos Q4
БС3
SJR0.153
CiteScore1.1
Impact factor0.5
ISSN00271314, 19350260
General Chemistry
Краткое описание
We study the effect of the nature of the substituent in the β-cyclodextrin derivative on the physicochemical properties of the antibacterial drug ciprofloxacin (CF). CF can form guest–host inclusion complexes with β-cyclodextrin derivatives, characterized by dissociation constants (Kdis) in the range of 10–3 to 10–4 M. A ligand with a small polar uncharged substituent (2-hydroxypropyl) form of the most stable complex, which also helps to increase the solubility of CF by 20 and 64% in buffer systems having a pH of 4.0 and 7.4, respectively. The inclusion of CF in a complex with Kdis = 10–3 M or lower contributes to a slower release of the drug. The physicochemical properties of the obtained complexes allow developing a highly effective formulation of the drug.
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Skuredina A. A. et al. Physical and Chemical Properties of the Guest–Host Inclusion Complexes of Cyprofloxacin with β-Cyclodextrin Derivatives // Moscow University Chemistry Bulletin. 2020. Vol. 75. No. 4. pp. 218-224.
ГОСТ со всеми авторами (до 50) Скопировать
Skuredina A. A., Kopnova T. Yu., Le Deygen I. M., Kudryashova E. V. Physical and Chemical Properties of the Guest–Host Inclusion Complexes of Cyprofloxacin with β-Cyclodextrin Derivatives // Moscow University Chemistry Bulletin. 2020. Vol. 75. No. 4. pp. 218-224.
RIS |
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TY - JOUR
DO - 10.3103/S0027131420040069
UR - https://doi.org/10.3103/S0027131420040069
TI - Physical and Chemical Properties of the Guest–Host Inclusion Complexes of Cyprofloxacin with β-Cyclodextrin Derivatives
T2 - Moscow University Chemistry Bulletin
AU - Skuredina, A A
AU - Kopnova, T Yu
AU - Le Deygen, I M
AU - Kudryashova, E V
PY - 2020
DA - 2020/07/01
PB - Pleiades Publishing
SP - 218-224
IS - 4
VL - 75
SN - 0027-1314
SN - 1935-0260
ER -
BibTex |
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@article{2020_Skuredina,
author = {A A Skuredina and T Yu Kopnova and I M Le Deygen and E V Kudryashova},
title = {Physical and Chemical Properties of the Guest–Host Inclusion Complexes of Cyprofloxacin with β-Cyclodextrin Derivatives},
journal = {Moscow University Chemistry Bulletin},
year = {2020},
volume = {75},
publisher = {Pleiades Publishing},
month = {jul},
url = {https://doi.org/10.3103/S0027131420040069},
number = {4},
pages = {218--224},
doi = {10.3103/S0027131420040069}
}
MLA
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Skuredina, A. A., et al. “Physical and Chemical Properties of the Guest–Host Inclusion Complexes of Cyprofloxacin with β-Cyclodextrin Derivatives.” Moscow University Chemistry Bulletin, vol. 75, no. 4, Jul. 2020, pp. 218-224. https://doi.org/10.3103/S0027131420040069.