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volume 2018 issue 1 pages M981

A Novel Disulfide-Containing Polycationic Amphiphile: 1,28-Di[(cholest-5-en-3β-yl)disulfanyl]-4,25-dioxo-3,8,12,17,21,26-hexaazaoctacosane Tetrahydrochloride

Publication typeJournal Article
Publication date2018-02-18
scimago Q4
wos Q4
SJR0.142
CiteScore0.9
Impact factor0.4
ISSN14228599
Organic Chemistry
Biochemistry
Physical and Theoretical Chemistry
Abstract

The absence of highly effective delivery systems is a major challenge for gene therapy. Our work was aimed at the development of novel cationic liposomes possessing high transfection efficiency. For this purpose, a novel disulfide polycationic amphiphile 2S4 was synthesized. Cationic liposomes based on 2S4 and a helper lipid DOPE were formed by the thin film hydration method and exhibited effective plasmid DNA delivery into the HEK293 cells, with a transfection activity superior to that of the commercial agent Lipofectamine® 2000. Our results suggest that the polycationic amphiphile 2S4 is a promising candidate for in vitro nucleic acid delivery.

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Puchkov P. A. et al. A Novel Disulfide-Containing Polycationic Amphiphile: 1,28-Di[(cholest-5-en-3β-yl)disulfanyl]-4,25-dioxo-3,8,12,17,21,26-hexaazaoctacosane Tetrahydrochloride // MolBank. 2018. Vol. 2018. No. 1. p. M981.
GOST all authors (up to 50) Copy
Puchkov P. A., Shmendel E. V., Andreeva V. D., Morozova N. G., Zenkova M. A., Maslov M. A., Maslov M. A Novel Disulfide-Containing Polycationic Amphiphile: 1,28-Di[(cholest-5-en-3β-yl)disulfanyl]-4,25-dioxo-3,8,12,17,21,26-hexaazaoctacosane Tetrahydrochloride // MolBank. 2018. Vol. 2018. No. 1. p. M981.
RIS |
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TY - JOUR
DO - 10.3390/M981
UR - https://www.mdpi.com/1422-8599/2018/1/M981
TI - A Novel Disulfide-Containing Polycationic Amphiphile: 1,28-Di[(cholest-5-en-3β-yl)disulfanyl]-4,25-dioxo-3,8,12,17,21,26-hexaazaoctacosane Tetrahydrochloride
T2 - MolBank
AU - Puchkov, Pavel A
AU - Shmendel, Elena V
AU - Andreeva, Valeria D
AU - Morozova, Nina G.
AU - Zenkova, Marina A
AU - Maslov, Mikhail A
AU - Maslov, Michael
PY - 2018
DA - 2018/02/18
PB - MDPI
SP - M981
IS - 1
VL - 2018
SN - 1422-8599
ER -
BibTex |
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BibTex (up to 50 authors) Copy
@article{2018_Puchkov,
author = {Pavel A Puchkov and Elena V Shmendel and Valeria D Andreeva and Nina G. Morozova and Marina A Zenkova and Mikhail A Maslov and Michael Maslov},
title = {A Novel Disulfide-Containing Polycationic Amphiphile: 1,28-Di[(cholest-5-en-3β-yl)disulfanyl]-4,25-dioxo-3,8,12,17,21,26-hexaazaoctacosane Tetrahydrochloride},
journal = {MolBank},
year = {2018},
volume = {2018},
publisher = {MDPI},
month = {feb},
url = {https://www.mdpi.com/1422-8599/2018/1/M981},
number = {1},
pages = {M981},
doi = {10.3390/M981}
}
MLA
Cite this
MLA Copy
Puchkov, Pavel A., et al. “A Novel Disulfide-Containing Polycationic Amphiphile: 1,28-Di[(cholest-5-en-3β-yl)disulfanyl]-4,25-dioxo-3,8,12,17,21,26-hexaazaoctacosane Tetrahydrochloride.” MolBank, vol. 2018, no. 1, Feb. 2018, p. M981. https://www.mdpi.com/1422-8599/2018/1/M981.