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volume 18 issue 2 pages 2096-2109

Palladium-catalyzed amination of dichloroquinolines with adamantane-containing amines

Publication typeJournal Article
Publication date2013-02-06
scimago Q1
wos Q2
SJR0.865
CiteScore8.6
Impact factor4.6
ISSN14203049
Organic Chemistry
Drug Discovery
Physical and Theoretical Chemistry
Pharmaceutical Science
Molecular Medicine
Analytical Chemistry
Chemistry (miscellaneous)
Abstract
Pd-catalyzed amination of isomeric 2,6-, 2,8-, 4,8- and 4,7-dichloroquinolines was studied using adamantane-containing amines in which substituents at the nitrogen atom differ in bulkiness. The selectivity of the amination of 2,6-dichloroquinoline was very low, substantially better results were obtained with 2,8-dichloroquinoline, and 4,8- and 4,7-dichloroquinolines provided the best yields of the amination products. Diamination of 4,8- and 4,7-dichloroquinolines was carried out with two amines which differ strongly in the bulkiness of the alkyl group. In the majority of cases BINAP ligand was successfully applied, however, it had to be replaced with DavePhos in certain reactions when using the most sterically hindered amine as well as for the diamination reactions.
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GOST Copy
Abel A. et al. Palladium-catalyzed amination of dichloroquinolines with adamantane-containing amines // Molecules. 2013. Vol. 18. No. 2. pp. 2096-2109.
GOST all authors (up to 50) Copy
Abel A., Averin A., Maloshitskaya O., Savelyev E., Orlinson B., Novakov I., Beletskaya I. Palladium-catalyzed amination of dichloroquinolines with adamantane-containing amines // Molecules. 2013. Vol. 18. No. 2. pp. 2096-2109.
RIS |
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RIS Copy
TY - JOUR
DO - 10.3390/molecules18022096
UR - https://doi.org/10.3390/molecules18022096
TI - Palladium-catalyzed amination of dichloroquinolines with adamantane-containing amines
T2 - Molecules
AU - Abel, Anton
AU - Averin, Alexei
AU - Maloshitskaya, Olga
AU - Savelyev, Evgenii
AU - Orlinson, Boris
AU - Novakov, Ivan
AU - Beletskaya, Irina
PY - 2013
DA - 2013/02/06
PB - MDPI
SP - 2096-2109
IS - 2
VL - 18
PMID - 23389254
SN - 1420-3049
ER -
BibTex |
Cite this
BibTex (up to 50 authors) Copy
@article{2013_Abel,
author = {Anton Abel and Alexei Averin and Olga Maloshitskaya and Evgenii Savelyev and Boris Orlinson and Ivan Novakov and Irina Beletskaya},
title = {Palladium-catalyzed amination of dichloroquinolines with adamantane-containing amines},
journal = {Molecules},
year = {2013},
volume = {18},
publisher = {MDPI},
month = {feb},
url = {https://doi.org/10.3390/molecules18022096},
number = {2},
pages = {2096--2109},
doi = {10.3390/molecules18022096}
}
MLA
Cite this
MLA Copy
Abel, Anton, et al. “Palladium-catalyzed amination of dichloroquinolines with adamantane-containing amines.” Molecules, vol. 18, no. 2, Feb. 2013, pp. 2096-2109. https://doi.org/10.3390/molecules18022096.