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volume 26 issue 24 pages 7493

Monoterpene-Containing Substituted Coumarins as Inhibitors of Respiratory Syncytial Virus (RSV) Replication

Publication typeJournal Article
Publication date2021-12-10
scimago Q1
wos Q2
SJR0.865
CiteScore8.6
Impact factor4.6
ISSN14203049
Organic Chemistry
Drug Discovery
Physical and Theoretical Chemistry
Pharmaceutical Science
Molecular Medicine
Analytical Chemistry
Chemistry (miscellaneous)
Abstract

Respiratory syncytial virus (RSV) is a critical cause of infant mortality. However, there are no vaccines and adequate drugs for its treatment. We showed, for the first time, that O-linked coumarin–monoterpene conjugates are effective RSV inhibitors. The most potent compounds are active against both RSV serotypes, A and B. According to the results of the time-of-addition experiment, the conjugates act at the early stages of virus cycle. Based on molecular modelling data, RSV F protein may be considered as a possible target.

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GOST |
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GOST Copy
Khomenko T. M. et al. Monoterpene-Containing Substituted Coumarins as Inhibitors of Respiratory Syncytial Virus (RSV) Replication // Molecules. 2021. Vol. 26. No. 24. p. 7493.
GOST all authors (up to 50) Copy
Khomenko T. M., Shtro A. A., Galochkina A. V., Nikolaeva Y. V., Petukhova G. D., Borisevich S. S., Korchagina D. V., Volcho K. P., Salakhutdinov N. F. Monoterpene-Containing Substituted Coumarins as Inhibitors of Respiratory Syncytial Virus (RSV) Replication // Molecules. 2021. Vol. 26. No. 24. p. 7493.
RIS |
Cite this
RIS Copy
TY - JOUR
DO - 10.3390/molecules26247493
UR - https://doi.org/10.3390/molecules26247493
TI - Monoterpene-Containing Substituted Coumarins as Inhibitors of Respiratory Syncytial Virus (RSV) Replication
T2 - Molecules
AU - Khomenko, Tatyana M
AU - Shtro, Anna A.
AU - Galochkina, Anastasia V.
AU - Nikolaeva, Yulia V
AU - Petukhova, Galina D
AU - Borisevich, Sophia S.
AU - Korchagina, Dina V.
AU - Volcho, Konstantin P.
AU - Salakhutdinov, Nariman F.
PY - 2021
DA - 2021/12/10
PB - MDPI
SP - 7493
IS - 24
VL - 26
PMID - 34946573
SN - 1420-3049
ER -
BibTex |
Cite this
BibTex (up to 50 authors) Copy
@article{2021_Khomenko,
author = {Tatyana M Khomenko and Anna A. Shtro and Anastasia V. Galochkina and Yulia V Nikolaeva and Galina D Petukhova and Sophia S. Borisevich and Dina V. Korchagina and Konstantin P. Volcho and Nariman F. Salakhutdinov},
title = {Monoterpene-Containing Substituted Coumarins as Inhibitors of Respiratory Syncytial Virus (RSV) Replication},
journal = {Molecules},
year = {2021},
volume = {26},
publisher = {MDPI},
month = {dec},
url = {https://doi.org/10.3390/molecules26247493},
number = {24},
pages = {7493},
doi = {10.3390/molecules26247493}
}
MLA
Cite this
MLA Copy
Khomenko, Tatyana M., et al. “Monoterpene-Containing Substituted Coumarins as Inhibitors of Respiratory Syncytial Virus (RSV) Replication.” Molecules, vol. 26, no. 24, Dec. 2021, p. 7493. https://doi.org/10.3390/molecules26247493.