A Photoswitchable Ligand Targeting the β 1 ‐Adrenoceptor Enables Light‐Control of the Cardiac Rhythm**

Anna Duran Corbera 1
Melissa Faria 2
Yuanyuan Ma 3
Eva Prats 4
Andre Dias 3
Juanlo Catena 5
Karen L Martinez 3
Demetrio Raldúa 2
Amadeu Llebaria 1
Xavier Rovira 1, 6
Publication typeJournal Article
Publication date2022-06-09
scimago Q1
wos Q1
SJR5.550
CiteScore27.6
Impact factor16.9
ISSN14337851, 15213773
General Chemistry
Catalysis
Abstract
New azobenzene-based molecular photoswitches active for the therapeutic β1-adrenoceptor (β1-AR) are presented. The most promising candidate, named pAzo-2, has a potency and β1/β2 selectivity similar to approved beta blockers. Importantly, pAzo-2 is compatible with imaging techniques and its potential as a cardioselective light-controlled drug has been validated by the reversible photomodulation of the cardiac rhythm in living zebrafish larvae.
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Duran Corbera A. et al. A Photoswitchable Ligand Targeting the β 1 ‐Adrenoceptor Enables Light‐Control of the Cardiac Rhythm** // Angewandte Chemie - International Edition. 2022. Vol. 61. No. 30.
GOST all authors (up to 50) Copy
Duran Corbera A., Faria M., Ma Y., Prats E., Dias A., Catena J., Martinez K. L., Raldúa D., Llebaria A., Rovira X. A Photoswitchable Ligand Targeting the β 1 ‐Adrenoceptor Enables Light‐Control of the Cardiac Rhythm** // Angewandte Chemie - International Edition. 2022. Vol. 61. No. 30.
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RIS Copy
TY - JOUR
DO - 10.1002/anie.202203449
UR - https://doi.org/10.1002/anie.202203449
TI - A Photoswitchable Ligand Targeting the β 1 ‐Adrenoceptor Enables Light‐Control of the Cardiac Rhythm**
T2 - Angewandte Chemie - International Edition
AU - Duran Corbera, Anna
AU - Faria, Melissa
AU - Ma, Yuanyuan
AU - Prats, Eva
AU - Dias, Andre
AU - Catena, Juanlo
AU - Martinez, Karen L
AU - Raldúa, Demetrio
AU - Llebaria, Amadeu
AU - Rovira, Xavier
PY - 2022
DA - 2022/06/09
PB - Wiley
IS - 30
VL - 61
PMID - 35608051
SN - 1433-7851
SN - 1521-3773
ER -
BibTex
Cite this
BibTex (up to 50 authors) Copy
@article{2022_Duran Corbera,
author = {Anna Duran Corbera and Melissa Faria and Yuanyuan Ma and Eva Prats and Andre Dias and Juanlo Catena and Karen L Martinez and Demetrio Raldúa and Amadeu Llebaria and Xavier Rovira},
title = {A Photoswitchable Ligand Targeting the β 1 ‐Adrenoceptor Enables Light‐Control of the Cardiac Rhythm**},
journal = {Angewandte Chemie - International Edition},
year = {2022},
volume = {61},
publisher = {Wiley},
month = {jun},
url = {https://doi.org/10.1002/anie.202203449},
number = {30},
doi = {10.1002/anie.202203449}
}