Chemistry of Heterocyclic Compounds

, volume 50 , issue 5 , pages 670-676

Synthesis and Intramolecular Cyclization of N-acyl- and N-allyl-N'-(2-oxo-1,2-dihydro-pyridin-3-yl)thiourea

I V Kulakov ¹

O S Nikitina ¹

A. S. Fisyuk ^{1, 2}

D S Goncharov ¹

Z T Shulgau ³

A E Gulyaev ³

Hide authors affiliations Show authors affiliations: 3 affiliations

F. M. Dostoevskii State University, Omsk, Russia |

Omsk State Technical University, Omsk, Russia |

Nazarbayev University, Center for Life Sciences, Astana, Kazakhstan |

Publication type: Journal Article

Publication date: 2014-07-13

Springer Nature

Chemistry of Heterocyclic Compounds

scimago Q4

wos Q4

SJR: 0.243

CiteScore: 2.7

Impact factor: 1.0

ISSN: 00093122, 15738353

DOI: 10.1007/s10593-014-1519-y

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Organic Chemistry

Abstract

The reaction of 3-amino-4,6-dimethylpyridin-2(1H)-one and 3-amino-4-phenylpyridin-2-one with acyl isothiocyanates (benzoyl-, 4-bromobenzoyl-, and methacryloyl isothiocyanates) and with allyl isothiocyanate has been studied. The N-carbamothioyl methacrylamides and N-allylthioureas obtained undergo intramolecular heterocyclization reactions to give the corresponding 1,3-thiazin-4-one and 1,3-thiazoline derivatives. It was found that the starting 3-amino-4,6-dimethylpyridin-2(1H)-one shows antiradical activity but the synthesized thioureas do not.

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9 citations

Palamarchuk Irina

23 publications, 160 citations

h-index: 8

University of Tyumen

3 citations

Shuvalov Vladislav

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PhD in Chemistry

24 publications, 147 citations

h-index: 8

Omsk State Technical University

Dostoevsky Omsk State University

Research interests

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1 citation

Vatsadze Sergey

DSc in Chemistry, professor, professor of the Russian Academy of Sciences

169 publications, 2 105 citations, 9 reviews

h-index: 20

N.D. Zelinsky Institute of Organic Chemistry of the Russian Academy of Sciences

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Supramolecular chemistry

1 citation

Fedorov Alexey

DSc in Chemistry, associate member of the Russian Academy of Sciences

93 publications, 2 829 citations, 10 reviews

h-index: 27

Lobachevsky State University of Nizhny Novgorod

1 citation

Novikov Mikhail

DSc in Chemistry, associate professor

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h-index: 33

Saint Petersburg State University

1 citation

Nyuchev Alexander

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PhD in Chemistry

43 publications, 1 267 citations, 27 reviews

h-index: 19

Lobachevsky State University of Nizhny Novgorod

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Flow Chemistry

Flow-through microreactors

1 citation

Zubkov Fedor

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DSc in Chemistry, professor

240 publications, 3 228 citations, 19 reviews

h-index: 31

Peoples' Friendship University of Russia

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Organic Chemistry

1 citation

Aksenov Aleksandr

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DSc in Chemistry, professor

244 publications, 2 194 citations, 15 reviews

h-index: 24

North Caucasus Federal University

Research interests

Medicinal Chemistry

Organic Chemistry

1 citation

Zakharova Lucia

DSc in Chemistry, professor

394 publications, 6 163 citations

h-index: 36

A.E. Arbuzov Institute of Organic and Physical Chemistry of the Kazan Scientific Center of the Russian Academy of Sciences

1 citation

Osyanin Vitaly

DSc in Chemistry, professor

131 publications, 1 144 citations, 3 reviews

h-index: 16

Samara State Technical University

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Organic Chemistry

1 citation

Tikhomirov Alexander

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60 publications, 927 citations

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Mendeleev University of Chemical Technology of Russia

Gause Institute of New Antibiotics

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Kulakov I. V. et al. Synthesis and Intramolecular Cyclization of N-acyl- and N-allyl-N'-(2-oxo-1,2-dihydro-pyridin-3-yl)thiourea // Chemistry of Heterocyclic Compounds. 2014. Vol. 50. No. 5. pp. 670-676.

GOST all authors (up to 50) Copy

Kulakov I. V., Nikitina O. S., Fisyuk A. S., Goncharov D. S., Shulgau Z. T., Gulyaev A. E. Synthesis and Intramolecular Cyclization of N-acyl- and N-allyl-N'-(2-oxo-1,2-dihydro-pyridin-3-yl)thiourea // Chemistry of Heterocyclic Compounds. 2014. Vol. 50. No. 5. pp. 670-676.

RIS |

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RIS Copy

TY - JOUR

DO - 10.1007/s10593-014-1519-y

UR - https://doi.org/10.1007/s10593-014-1519-y

TI - Synthesis and Intramolecular Cyclization of N-acyl- and N-allyl-N'-(2-oxo-1,2-dihydro-pyridin-3-yl)thiourea

T2 - Chemistry of Heterocyclic Compounds

AU - Kulakov, I V

AU - Nikitina, O S

AU - Fisyuk, A. S.

AU - Goncharov, D S

AU - Shulgau, Z T

AU - Gulyaev, A E

PY - 2014

DA - 2014/07/13

PB - Springer Nature

SP - 670-676

IS - 5

VL - 50

SN - 0009-3122

SN - 1573-8353

ER -

BibTex |

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BibTex (up to 50 authors) Copy

@article{2014_Kulakov,

author = {I V Kulakov and O S Nikitina and A. S. Fisyuk and D S Goncharov and Z T Shulgau and A E Gulyaev},

title = {Synthesis and Intramolecular Cyclization of N-acyl- and N-allyl-N'-(2-oxo-1,2-dihydro-pyridin-3-yl)thiourea},

journal = {Chemistry of Heterocyclic Compounds},

year = {2014},

volume = {50},

publisher = {Springer Nature},

month = {jul},

url = {https://doi.org/10.1007/s10593-014-1519-y},

number = {5},

pages = {670--676},

doi = {10.1007/s10593-014-1519-y}

}

MLA

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MLA Copy

Kulakov, I. V., et al. “Synthesis and Intramolecular Cyclization of N-acyl- and N-allyl-N'-(2-oxo-1,2-dihydro-pyridin-3-yl)thiourea.” Chemistry of Heterocyclic Compounds, vol. 50, no. 5, Jul. 2014, pp. 670-676. https://doi.org/10.1007/s10593-014-1519-y.