Synthesis of and HIV-1 Integrase Inhibition by 2-[7-(Fluorobenzyloxy)-4-Oxo-4hchromen-3-Yl]-1-Hydroxyimidazoles
Publication type: Journal Article
Publication date: 2016-11-19
scimago Q4
wos Q4
SJR: 0.219
CiteScore: 1.4
Impact factor: 1.0
ISSN: 0091150X, 15739031
Drug Discovery
Pharmacology
Abstract
A series of six new 2-[7-(fluorobenzyloxy)-4-oxo-4H-chromen-3-yl]-1-hydroxyimidazoles were synthesized and characterized as potential HIV-1 integrase inhibitors. Prototropic tautomerism of the obtained 1-hydroxyimidazoles was discussed. Their ability to inhibit integrase catalytic activity in 3′-terminal processing and chain transfer reactions was studied. It was shown that these compounds did not exhibit noticeable inhibition.
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Total citations:
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Citations from 2024:
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(33.34%)
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Nikitina P. A. et al. Synthesis of and HIV-1 Integrase Inhibition by 2-[7-(Fluorobenzyloxy)-4-Oxo-4hchromen-3-Yl]-1-Hydroxyimidazoles // Pharmaceutical Chemistry Journal. 2016. Vol. 50. No. 8. pp. 513-518.
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Nikitina P. A., Tkach I. I., Knyazhanskaya E. S., Gottikh M. B., Perevalov V. P. Synthesis of and HIV-1 Integrase Inhibition by 2-[7-(Fluorobenzyloxy)-4-Oxo-4hchromen-3-Yl]-1-Hydroxyimidazoles // Pharmaceutical Chemistry Journal. 2016. Vol. 50. No. 8. pp. 513-518.
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TY - JOUR
DO - 10.1007/s11094-016-1479-x
UR - https://doi.org/10.1007/s11094-016-1479-x
TI - Synthesis of and HIV-1 Integrase Inhibition by 2-[7-(Fluorobenzyloxy)-4-Oxo-4hchromen-3-Yl]-1-Hydroxyimidazoles
T2 - Pharmaceutical Chemistry Journal
AU - Nikitina, P A
AU - Tkach, I. I.
AU - Knyazhanskaya, E S
AU - Gottikh, M B
AU - Perevalov, V P
PY - 2016
DA - 2016/11/19
PB - Springer Nature
SP - 513-518
IS - 8
VL - 50
SN - 0091-150X
SN - 1573-9031
ER -
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BibTex (up to 50 authors)
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@article{2016_Nikitina,
author = {P A Nikitina and I. I. Tkach and E S Knyazhanskaya and M B Gottikh and V P Perevalov},
title = {Synthesis of and HIV-1 Integrase Inhibition by 2-[7-(Fluorobenzyloxy)-4-Oxo-4hchromen-3-Yl]-1-Hydroxyimidazoles},
journal = {Pharmaceutical Chemistry Journal},
year = {2016},
volume = {50},
publisher = {Springer Nature},
month = {nov},
url = {https://doi.org/10.1007/s11094-016-1479-x},
number = {8},
pages = {513--518},
doi = {10.1007/s11094-016-1479-x}
}
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MLA
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Nikitina, P. A., et al. “Synthesis of and HIV-1 Integrase Inhibition by 2-[7-(Fluorobenzyloxy)-4-Oxo-4hchromen-3-Yl]-1-Hydroxyimidazoles.” Pharmaceutical Chemistry Journal, vol. 50, no. 8, Nov. 2016, pp. 513-518. https://doi.org/10.1007/s11094-016-1479-x.