Chemistry of Heterocyclic Compounds, volume 56, issue 6, pages 756-762

Structure and antibacterial activity (mediated by the SOS response) of spiropiperidinium salts obtained by cyclization of Mannich bases of arylaliphatic 1,5-diketones

Bukreev Aleksey V ¹

Akimova Taisia I ¹

Osterman Ilya А ^{2, 3}

Shakhtina Anna N ³

Khudyakova Yuliya V ⁴

Gerasimenko Andrey V ⁵

Sergiev Petr V. ^{2, 3}

Dontsova Olga А ^{2, 3, 6}

Deryabin Pavel I ¹

Kolycheva Vera B ¹

Hide authors affiliations Show authors affiliations: 6 affiliations

Far Eastern Federal University, School of Natural Sciences, Vladivostok, Russia |

Skolkovo Institute of Science and Technology, Center of Life Sciences, Moscow, Russia |

Lomonosov Moscow state University, Moscow, Russia |

⁴

G. B. Elyakov Pacific Institute of Bioorganic Chemistry, Vladivostok, Russia |

⁵

Institute of Chemistry, Far Eastern Branch of the Russian Academy of Sciences, Vladivostok, Russia |

⁶

Shemyakin-Ovchinnikov Institute of Bioorganic Chemistry, Russian Academy of Sciences, Moscow, Russia |

Publication type: Journal Article

Publication date: 2020-06-01

Springer Nature

Journal: Chemistry of Heterocyclic Compounds

Quartile SCImago

Quartile WOS

Impact factor: 1.5

ISSN: 00093122, 15738353

DOI: 10.1007/s10593-020-02727-z

Copy DOI

Organic Chemistry

Abstract

New derivatives of 3,5-dibenzoylspiropiperidinium salts were obtained by the previously developed method of cyclization of Mannich methylidene monobases of arylaliphatic 1,5-diketones and their antibacterial activity was studied. The structure of one of the salts was determined by X-ray structural analysis. The study of the mechanism of action using the pDualrep2 reporter system showed that some compounds cause the SOS response in the bacterial cell.

By date By citations

Citations by journals

	1
Journal of Organic Chemistry	Journal of Organic Chemistry, 1, 100% Journal of Organic Chemistry 1 publication, 100%
	1

Citations by publishers

	1
American Chemical Society (ACS)	American Chemical Society (ACS), 1, 100% American Chemical Society (ACS) 1 publication, 100%
	1

We do not take into account publications that without a DOI.
Statistics recalculated only for publications connected to researchers, organizations and labs registered on the platform.
Statistics recalculated weekly.

{"yearsCitations":{"type":"bar","data":{"show":true,"labels":[2022],"ids":[0],"codes":[0],"imageUrls":[""],"datasets":[{"label":"Citations number","data":[1],"backgroundColor":["#3B82F6"],"percentage":["100"],"barThickness":null}]},"options":{"indexAxis":"x","maintainAspectRatio":true,"scales":{"y":{"ticks":{"precision":0,"autoSkip":false,"font":{"family":"Montserrat"},"color":"#000000"}},"x":{"ticks":{"stepSize":1,"precision":0,"font":{"family":"Montserrat"},"color":"#000000"}}},"plugins":{"legend":{"position":"top","labels":{"font":{"family":"Montserrat"},"color":"#000000"}},"title":{"display":true,"text":"Citations per year","font":{"size":24,"family":"Montserrat","weight":600},"color":"#000000"}}}},"journals":{"type":"bar","data":{"show":true,"labels":["Journal of Organic Chemistry"],"ids":[8697],"codes":[0],"imageUrls":["\/storage\/images\/resized\/iLiQsFqFaSEx6chlGQ5fbAwF6VYU3WWa08hkss0g_medium.webp"],"datasets":[{"label":"","data":[1],"backgroundColor":["#3B82F6"],"percentage":[100],"barThickness":13}]},"options":{"indexAxis":"y","maintainAspectRatio":false,"scales":{"y":{"ticks":{"precision":0,"autoSkip":false,"font":{"family":"Montserrat"},"color":"#000000"}},"x":{"ticks":{"stepSize":null,"precision":0,"font":{"family":"Montserrat"},"color":"#000000"}}},"plugins":{"legend":{"position":"top","labels":{"font":{"family":"Montserrat"},"color":"#000000"}},"title":{"display":true,"text":"Journals","font":{"size":24,"family":"Montserrat","weight":600},"color":"#000000"}}}},"publishers":{"type":"bar","data":{"show":true,"labels":["American Chemical Society (ACS)"],"ids":[40],"codes":[0],"imageUrls":["\/storage\/images\/resized\/iLiQsFqFaSEx6chlGQ5fbAwF6VYU3WWa08hkss0g_medium.webp"],"datasets":[{"label":"","data":[1],"backgroundColor":["#3B82F6"],"percentage":[100],"barThickness":13}]},"options":{"indexAxis":"y","maintainAspectRatio":false,"scales":{"y":{"ticks":{"precision":0,"autoSkip":false,"font":{"family":"Montserrat"},"color":"#000000"}},"x":{"ticks":{"stepSize":null,"precision":0,"font":{"family":"Montserrat"},"color":"#000000"}}},"plugins":{"legend":{"position":"top","labels":{"font":{"family":"Montserrat"},"color":"#000000"}},"title":{"display":true,"text":"Publishers","font":{"size":24,"family":"Montserrat","weight":600},"color":"#000000"}}}}}

Metrics

Cite this

GOST |

Cite this

GOST Copy

Bukreev A. V. et al. Structure and antibacterial activity (mediated by the SOS response) of spiropiperidinium salts obtained by cyclization of Mannich bases of arylaliphatic 1,5-diketones // Chemistry of Heterocyclic Compounds. 2020. Vol. 56. No. 6. pp. 756-762.

GOST all authors (up to 50) Copy

Bukreev A. V., Akimova T. I., Osterman I. А., Shakhtina A. N., Khudyakova Y. V., Gerasimenko A. V., Sergiev P. V., Dontsova O. А., Deryabin P. I., Kolycheva V. B. Structure and antibacterial activity (mediated by the SOS response) of spiropiperidinium salts obtained by cyclization of Mannich bases of arylaliphatic 1,5-diketones // Chemistry of Heterocyclic Compounds. 2020. Vol. 56. No. 6. pp. 756-762.

RIS |

Cite this

RIS Copy

TY - JOUR

DO - 10.1007/s10593-020-02727-z

UR - https://doi.org/10.1007%2Fs10593-020-02727-z

TI - Structure and antibacterial activity (mediated by the SOS response) of spiropiperidinium salts obtained by cyclization of Mannich bases of arylaliphatic 1,5-diketones

T2 - Chemistry of Heterocyclic Compounds

AU - Bukreev, Aleksey V

AU - Akimova, Taisia I

AU - Osterman, Ilya А

AU - Shakhtina, Anna N

AU - Khudyakova, Yuliya V

AU - Gerasimenko, Andrey V

AU - Sergiev, Petr V.

AU - Dontsova, Olga А

AU - Deryabin, Pavel I

AU - Kolycheva, Vera B

PY - 2020

DA - 2020/06/01 00:00:00

PB - Springer Nature

SP - 756-762

IS - 6

VL - 56

SN - 0009-3122

SN - 1573-8353

ER -

BibTex |

Cite this

BibTex Copy

@article{2020_Bukreev,

author = {Aleksey V Bukreev and Taisia I Akimova and Ilya А Osterman and Anna N Shakhtina and Yuliya V Khudyakova and Andrey V Gerasimenko and Petr V. Sergiev and Olga А Dontsova and Pavel I Deryabin and Vera B Kolycheva},

title = {Structure and antibacterial activity (mediated by the SOS response) of spiropiperidinium salts obtained by cyclization of Mannich bases of arylaliphatic 1,5-diketones},

journal = {Chemistry of Heterocyclic Compounds},

year = {2020},

volume = {56},

publisher = {Springer Nature},

month = {jun},

url = {https://doi.org/10.1007%2Fs10593-020-02727-z},

number = {6},

pages = {756--762},

doi = {10.1007/s10593-020-02727-z}

}

MLA

Cite this

MLA Copy

Bukreev, Aleksey V., et al. “Structure and antibacterial activity (mediated by the SOS response) of spiropiperidinium salts obtained by cyclization of Mannich bases of arylaliphatic 1,5-diketones.” Chemistry of Heterocyclic Compounds, vol. 56, no. 6, Jun. 2020, pp. 756-762. https://doi.org/10.1007%2Fs10593-020-02727-z.

Found error?

Publisher

Springer Nature

Journal

Chemistry of Heterocyclic Compounds

Quartile SCImago

Quartile WOS

Impact factor

1.5

ISSN

00093122 (Print)
15738353 (Electronic)

Labs

Laboratory of Nucleoprotein Chemistry, Department of Chemistry of Natural Compounds, Faculty of Chemistry

Profiles