Pharmaceutical Chemistry Journal, volume 53, issue 4, pages 288-297
Conjugates of Prostate-Specific Membrane Antigen Ligands with Antitumor Drugs
Publication type: Journal Article
Publication date: 2019-07-09
Journal:
Pharmaceutical Chemistry Journal
Quartile SCImago
Q4
Quartile WOS
Q4
Impact factor: 0.9
ISSN: 0091150X, 15739031
Drug Discovery
Pharmacology
Abstract
Conjugates for targeted delivery that are based on low-molecular-mass prostate specific membrane antigen (PSMA) inhibitors are widely used and developed because of the deficiencies of existing methods for treating and diagnosing prostate cancer. The major classes of low-molecular-mass PSMA inhibitors, drug classes, and their mechanisms of action are discussed. Therapeutic conjugates for targeted delivery that are based on them are analyzed. Structural features of the linker that affect the biological activity and selectivity are identified.
Citations by journals
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Mendeleev Communications
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Mendeleev Communications
1 publication, 50%
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Molecules
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Molecules
1 publication, 50%
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1
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Citations by publishers
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1
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Elsevier
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Elsevier
1 publication, 50%
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Multidisciplinary Digital Publishing Institute (MDPI)
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Multidisciplinary Digital Publishing Institute (MDPI)
1 publication, 50%
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1
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GOST
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Uspenskaya A. A. et al. Conjugates of Prostate-Specific Membrane Antigen Ligands with Antitumor Drugs // Pharmaceutical Chemistry Journal. 2019. Vol. 53. No. 4. pp. 288-297.
GOST all authors (up to 50)
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Uspenskaya A. A., Machulkin A. E., Mazhuga A. G., Beloglazkina E. K. Conjugates of Prostate-Specific Membrane Antigen Ligands with Antitumor Drugs // Pharmaceutical Chemistry Journal. 2019. Vol. 53. No. 4. pp. 288-297.
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RIS
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TY - JOUR
DO - 10.1007/s11094-019-01994-1
UR - https://doi.org/10.1007%2Fs11094-019-01994-1
TI - Conjugates of Prostate-Specific Membrane Antigen Ligands with Antitumor Drugs
T2 - Pharmaceutical Chemistry Journal
AU - Uspenskaya, A A
AU - Machulkin, A E
AU - Mazhuga, A G
AU - Beloglazkina, E K
PY - 2019
DA - 2019/07/09 00:00:00
PB - Springer Nature
SP - 288-297
IS - 4
VL - 53
SN - 0091-150X
SN - 1573-9031
ER -
Cite this
BibTex
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@article{2019_Uspenskaya,
author = {A A Uspenskaya and A E Machulkin and A G Mazhuga and E K Beloglazkina},
title = {Conjugates of Prostate-Specific Membrane Antigen Ligands with Antitumor Drugs},
journal = {Pharmaceutical Chemistry Journal},
year = {2019},
volume = {53},
publisher = {Springer Nature},
month = {jul},
url = {https://doi.org/10.1007%2Fs11094-019-01994-1},
number = {4},
pages = {288--297},
doi = {10.1007/s11094-019-01994-1}
}
Cite this
MLA
Copy
Uspenskaya, A. A., et al. “Conjugates of Prostate-Specific Membrane Antigen Ligands with Antitumor Drugs.” Pharmaceutical Chemistry Journal, vol. 53, no. 4, Jul. 2019, pp. 288-297. https://doi.org/10.1007%2Fs11094-019-01994-1.