First total synthesis of aerucyclamide B
Publication type: Journal Article
Publication date: 2013-05-01
scimago Q3
wos Q3
SJR: 0.334
CiteScore: 3.2
Impact factor: 1.5
ISSN: 00404039, 18733581
Organic Chemistry
Drug Discovery
Biochemistry
Abstract
The first total synthesis of the antimalarial aerucyclamide B has been achieved in 9% overall yield. Two thiazoles and a dipeptide were used to prepare two open precursors of cyclo-Gly-l-allo-Thr-l-Ile-Thz-d-allo-Ile-Thz. Cyclodehydration with Deoxo-Fluor of the β-hydroxyamide present in the macrocycle, rendered aerucyclamide B (67%) and an unexpected fluorous derivative (28%).
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Total citations:
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Citations from 2024:
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GOST
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Peña S. et al. First total synthesis of aerucyclamide B // Tetrahedron Letters. 2013. Vol. 54. No. 22. pp. 2806-2808.
GOST all authors (up to 50)
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Peña S., Scarone L., Manta E., Serra G. L. First total synthesis of aerucyclamide B // Tetrahedron Letters. 2013. Vol. 54. No. 22. pp. 2806-2808.
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RIS
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TY - JOUR
DO - 10.1016/j.tetlet.2013.03.060
UR - https://doi.org/10.1016/j.tetlet.2013.03.060
TI - First total synthesis of aerucyclamide B
T2 - Tetrahedron Letters
AU - Peña, Stella
AU - Scarone, Laura
AU - Manta, Eduardo
AU - Serra, Gloria L
PY - 2013
DA - 2013/05/01
PB - Elsevier
SP - 2806-2808
IS - 22
VL - 54
SN - 0040-4039
SN - 1873-3581
ER -
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BibTex (up to 50 authors)
Copy
@article{2013_Peña,
author = {Stella Peña and Laura Scarone and Eduardo Manta and Gloria L Serra},
title = {First total synthesis of aerucyclamide B},
journal = {Tetrahedron Letters},
year = {2013},
volume = {54},
publisher = {Elsevier},
month = {may},
url = {https://doi.org/10.1016/j.tetlet.2013.03.060},
number = {22},
pages = {2806--2808},
doi = {10.1016/j.tetlet.2013.03.060}
}
Cite this
MLA
Copy
Peña, Stella, et al. “First total synthesis of aerucyclamide B.” Tetrahedron Letters, vol. 54, no. 22, May. 2013, pp. 2806-2808. https://doi.org/10.1016/j.tetlet.2013.03.060.