The synthesis and antituberculosis activity of 5'-nor carbocyclic uracil derivatives.
Тип публикации: Journal Article
Дата публикации: 2012-11-01
scimago Q2
wos Q1
БС1
SJR: 0.608
CiteScore: 6.7
Impact factor: 3.0
ISSN: 09680896, 14643391
PubMed ID:
23062712
Organic Chemistry
Drug Discovery
Biochemistry
Molecular Biology
Pharmaceutical Science
Clinical Biochemistry
Molecular Medicine
Краткое описание
A series of new carbocyclic uracil derivatives were synthesized and evaluated as potential antituberculosis agents. Racemic 1-[4'-hydroxy-2'-cyclopenten-1'-yl]-5-tetradecynyluracil completely inhibited the growth of Mycobacterium tuberculosis H37Rv in vitro at a concentration of 10 μg/ml. Individual (+) and (-) isomers of the above uracil derivative were isolated and showed the same level of activity against two strains of Mycobacterium tuberculosis: laboratory sensitive (H37Rv) and clinical resistant to five top antituberculosis drugs (MS-115).
Найдено
Ничего не найдено, попробуйте изменить настройки фильтра.
Найдено
Ничего не найдено, попробуйте изменить настройки фильтра.
Топ-30
Журналы
|
1
2
3
4
5
6
7
|
|
|
Molecules
7 публикаций, 14.58%
|
|
|
Russian Journal of Bioorganic Chemistry
3 публикации, 6.25%
|
|
|
Russian Chemical Bulletin
3 публикации, 6.25%
|
|
|
Bioorganic and Medicinal Chemistry Letters
3 публикации, 6.25%
|
|
|
Bioorganic and Medicinal Chemistry
2 публикации, 4.17%
|
|
|
European Journal of Medicinal Chemistry
2 публикации, 4.17%
|
|
|
MedChemComm
2 публикации, 4.17%
|
|
|
Heterocyclic Communications
2 публикации, 4.17%
|
|
|
Mendeleev Communications
1 публикация, 2.08%
|
|
|
Russian Chemical Reviews
1 публикация, 2.08%
|
|
|
Biochimie
1 публикация, 2.08%
|
|
|
Journal of Antibiotics
1 публикация, 2.08%
|
|
|
Molecular Biology
1 публикация, 2.08%
|
|
|
Chemical Biology and Drug Design
1 публикация, 2.08%
|
|
|
Acta Naturae
1 публикация, 2.08%
|
|
|
Microorganisms
1 публикация, 2.08%
|
|
|
Future Medicinal Chemistry
1 публикация, 2.08%
|
|
|
Monatshefte fur Chemie
1 публикация, 2.08%
|
|
|
Journal of Chemical Crystallography
1 публикация, 2.08%
|
|
|
Medicinal Chemistry Research
1 публикация, 2.08%
|
|
|
Tetrahedron Letters
1 публикация, 2.08%
|
|
|
ChemMedChem
1 публикация, 2.08%
|
|
|
Nucleosides, Nucleotides and Nucleic Acids
1 публикация, 2.08%
|
|
|
Journal of Receptor and Signal Transduction Research
1 публикация, 2.08%
|
|
|
Pharmaceutical Chemistry Journal
1 публикация, 2.08%
|
|
|
Bulletin of Russian State Medical University
1 публикация, 2.08%
|
|
|
Annual Reports in Medicinal Chemistry
1 публикация, 2.08%
|
|
|
International Journal of Molecular Sciences
1 публикация, 2.08%
|
|
|
Current Organic Chemistry
1 публикация, 2.08%
|
|
|
Pharmaceutics
1 публикация, 2.08%
|
|
|
1
2
3
4
5
6
7
|
Издатели
|
2
4
6
8
10
|
|
|
Elsevier
10 публикаций, 20.83%
|
|
|
MDPI
10 публикаций, 20.83%
|
|
|
Springer Nature
9 публикаций, 18.75%
|
|
|
Pleiades Publishing
4 публикации, 8.33%
|
|
|
Taylor & Francis
3 публикации, 6.25%
|
|
|
Royal Society of Chemistry (RSC)
2 публикации, 4.17%
|
|
|
Wiley
2 публикации, 4.17%
|
|
|
Walter de Gruyter
2 публикации, 4.17%
|
|
|
OOO Zhurnal "Mendeleevskie Soobshcheniya"
1 публикация, 2.08%
|
|
|
Autonomous Non-profit Organization Editorial Board of the journal Uspekhi Khimii
1 публикация, 2.08%
|
|
|
Acta Naturae Ltd
1 публикация, 2.08%
|
|
|
Pirogov Russian National Research Medical University
1 публикация, 2.08%
|
|
|
Bentham Science Publishers Ltd.
1 публикация, 2.08%
|
|
|
A and V Publications
1 публикация, 2.08%
|
|
|
2
4
6
8
10
|
- Мы не учитываем публикации, у которых нет DOI.
- Статистика публикаций обновляется еженедельно.
Вы ученый?
Создайте профиль, чтобы получать персональные рекомендации коллег, конференций и новых статей.
Метрики
48
Всего цитирований:
48
Цитирований c 2025:
1
(2.08%)
Цитировать
ГОСТ |
RIS |
BibTex |
MLA
Цитировать
ГОСТ
Скопировать
Matyugina E. et al. The synthesis and antituberculosis activity of 5'-nor carbocyclic uracil derivatives. // Bioorganic and Medicinal Chemistry. 2012. Vol. 20. No. 22. pp. 6680-6686.
ГОСТ со всеми авторами (до 50)
Скопировать
Matyugina E., Khandazhinskaya A., Chernousova L., Andreevskaya S., Smirnova T., Chizhov A. O., Карпенко И. Л., Кочетков С. Н., Alexandrova L. The synthesis and antituberculosis activity of 5'-nor carbocyclic uracil derivatives. // Bioorganic and Medicinal Chemistry. 2012. Vol. 20. No. 22. pp. 6680-6686.
Цитировать
RIS
Скопировать
TY - JOUR
DO - 10.1016/j.bmc.2012.09.019
UR - https://doi.org/10.1016/j.bmc.2012.09.019
TI - The synthesis and antituberculosis activity of 5'-nor carbocyclic uracil derivatives.
T2 - Bioorganic and Medicinal Chemistry
AU - Matyugina, Elena
AU - Khandazhinskaya, Anastasia
AU - Chernousova, Larisa
AU - Andreevskaya, Sofia
AU - Smirnova, Tatiana
AU - Chizhov, A. O.
AU - Карпенко, И. Л.
AU - Кочетков, С. Н.
AU - Alexandrova, Ludmila
PY - 2012
DA - 2012/11/01
PB - Elsevier
SP - 6680-6686
IS - 22
VL - 20
PMID - 23062712
SN - 0968-0896
SN - 1464-3391
ER -
Цитировать
BibTex (до 50 авторов)
Скопировать
@article{2012_Matyugina,
author = {Elena Matyugina and Anastasia Khandazhinskaya and Larisa Chernousova and Sofia Andreevskaya and Tatiana Smirnova and A. O. Chizhov and И. Л. Карпенко and С. Н. Кочетков and Ludmila Alexandrova},
title = {The synthesis and antituberculosis activity of 5'-nor carbocyclic uracil derivatives.},
journal = {Bioorganic and Medicinal Chemistry},
year = {2012},
volume = {20},
publisher = {Elsevier},
month = {nov},
url = {https://doi.org/10.1016/j.bmc.2012.09.019},
number = {22},
pages = {6680--6686},
doi = {10.1016/j.bmc.2012.09.019}
}
Цитировать
MLA
Скопировать
Matyugina, Elena, et al. “The synthesis and antituberculosis activity of 5'-nor carbocyclic uracil derivatives..” Bioorganic and Medicinal Chemistry, vol. 20, no. 22, Nov. 2012, pp. 6680-6686. https://doi.org/10.1016/j.bmc.2012.09.019.