Bioorganic and Medicinal Chemistry

, volume 25 , issue 21 , pages 5891-5903

Recently reported biological activities of pyrazole compounds

Jessica Venancia Faria ^{1, 2}

Percilene Fazolin Vegi ²

Ana Gabriella Carvalho Miguita ³

Maurício C. dos Santos ³

Núbia Boechat ¹

Alice M. R. Bernardino ²

Hide authors affiliations Show authors affiliations: 3 affiliations

Fundação Oswaldo Cruz – Fiocruz, Instituto de Tecnologia em Fármacos – Farmanguinhos, Manguinhos, RJ, Brazil |

Programa de Pós-Graduação em Química,Instituto de Química, Universidade Federal Fluminense, Niterói, RJ, Brazil |

Laboratório de Síntese Orgânica (LABSINTO), Instituto de Física e Química, Universidade Federal de Itajubá, Itajubá, MG, Brazil |

Publication type: Journal Article

Publication date: 2017-11-01

Elsevier

Bioorganic and Medicinal Chemistry

scimago Q2

wos Q1

SJR: 0.608

CiteScore: 6.7

Impact factor: 3.0

ISSN: 09680896, 14643391

DOI: 10.1016/j.bmc.2017.09.035

Copy DOI

PubMed ID: 28988624

Organic Chemistry

Drug Discovery

Biochemistry

Molecular Biology

Pharmaceutical Science

Clinical Biochemistry

Molecular Medicine

Abstract

The pyrazole nucleus is an aromatic azole heterocycle with two adjacent nitrogen atoms. Pyrazole derivatives have exhibited a broad spectrum of biological activities, and approved pyrazole-containing drugs include celecoxib, antipyrine, phenylbutazone, rimonabant, and dipyrone. Many research groups have synthesized and evaluated pyrazoles against several biological agents. This review examines recent publications relating the structures of pyrazoles with their corresponding biological activities.

Found

2 citations

Shul'ts Elvira

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N.N. Vorozhtsov Novosibirsk Institute of Organic Chemistry of the Siberian Branch of the Russian Academy of Sciences

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Burmistrov Vladimir

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N.N. Vorozhtsov Novosibirsk Institute of Organic Chemistry of the Siberian Branch of the Russian Academy of Sciences

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Herzen State Pedagogical University of Russia

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Perm National Research Polytechnic University

Institute of Ecology and Genetics of Microorganisms of the Ural Branch of the Russian Academy of Sciences

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Antioxidants

Microbiology

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Dilman Alexander

DSc in Chemistry, associate member of the Russian Academy of Sciences

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N.D. Zelinsky Institute of Organic Chemistry of the Russian Academy of Sciences

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Library for Natural Sciences of the Russian Academy of Sciences

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Volgograd State Technical University

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Egyptian Atomic Energy Authority

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GOST |

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GOST Copy

Faria J. V. et al. Recently reported biological activities of pyrazole compounds // Bioorganic and Medicinal Chemistry. 2017. Vol. 25. No. 21. pp. 5891-5903.

GOST all authors (up to 50) Copy

Faria J. V., Vegi P. F., Miguita A. G. C., dos Santos M. C., Boechat N., Bernardino A. M. R. Recently reported biological activities of pyrazole compounds // Bioorganic and Medicinal Chemistry. 2017. Vol. 25. No. 21. pp. 5891-5903.

RIS |

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RIS Copy

TY - JOUR

DO - 10.1016/j.bmc.2017.09.035

UR - https://doi.org/10.1016/j.bmc.2017.09.035

TI - Recently reported biological activities of pyrazole compounds

T2 - Bioorganic and Medicinal Chemistry

AU - Faria, Jessica Venancia

AU - Vegi, Percilene Fazolin

AU - Miguita, Ana Gabriella Carvalho

AU - dos Santos, Maurício C.

AU - Boechat, Núbia

AU - Bernardino, Alice M. R.

PY - 2017

DA - 2017/11/01

PB - Elsevier

SP - 5891-5903

IS - 21

VL - 25

PMID - 28988624

SN - 0968-0896

SN - 1464-3391

ER -

BibTex |

Cite this

BibTex (up to 50 authors) Copy

@article{2017_Faria,

author = {Jessica Venancia Faria and Percilene Fazolin Vegi and Ana Gabriella Carvalho Miguita and Maurício C. dos Santos and Núbia Boechat and Alice M. R. Bernardino},

title = {Recently reported biological activities of pyrazole compounds},

journal = {Bioorganic and Medicinal Chemistry},

year = {2017},

volume = {25},

publisher = {Elsevier},

month = {nov},

url = {https://doi.org/10.1016/j.bmc.2017.09.035},

number = {21},

pages = {5891--5903},

doi = {10.1016/j.bmc.2017.09.035}

}

MLA

Cite this

MLA Copy

Faria, Jessica Venancia, et al. “Recently reported biological activities of pyrazole compounds.” Bioorganic and Medicinal Chemistry, vol. 25, no. 21, Nov. 2017, pp. 5891-5903. https://doi.org/10.1016/j.bmc.2017.09.035.

Publisher

Elsevier

Journal

Bioorganic and Medicinal Chemistry

scimago Q2

wos Q1

SJR

0.608

CiteScore

6.7

Impact factor

3.0

ISSN

09680896 (Print)

14643391 (Electronic)