Mendeleev Communications, volume 30, issue 6, pages 756-759
Influence of the dipeptide linker configuration on the activity of PSMA ligands
Beloglazkina Elena K
,
Nimenko Ekaterina A.
1
,
Majouga Alexander G.
,
Petrov Stanislav A
,
Shafikov Radik R
,
Skvortsov Dmitry A.
,
Machulkin Alexey E.
1
,
Shafikov Radik R
2
,
Skvortsov Dmitry
2
,
Majouga Alexander G.
3, 4
1
3
Publication type: Journal Article
Publication date: 2020-11-01
Journal:
Mendeleev Communications
Quartile SCImago
Q3
Quartile WOS
Q3
Impact factor: 1.9
ISSN: 09599436, 1364551X
General Chemistry
Abstract
Selective ligands of an urea-based prostate specific membrane antigen with a phenylalanine/tyrosine-based dipeptide linker and with a mingled chiral centers configuration and/or substituted aromatic fragments were prepared in seven steps by liquid- and in six steps by solid-phase synthesis. In vitro test for inhibiting the cleavage of N-acetylaspartylglutamate revealed the optimum linker containing l -phenylalanine in the structure on the N-terminus of a dipeptide chain.
Citations by journals
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1
2
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International Journal of Molecular Sciences
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International Journal of Molecular Sciences
2 publications, 40%
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Journal of Molecular Structure
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Journal of Molecular Structure
1 publication, 20%
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Bioorganic and Medicinal Chemistry Letters
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Bioorganic and Medicinal Chemistry Letters
1 publication, 20%
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Mendeleev Communications
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Mendeleev Communications
1 publication, 20%
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1
2
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Citations by publishers
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1
2
3
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Elsevier
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Elsevier
3 publications, 60%
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Multidisciplinary Digital Publishing Institute (MDPI)
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Multidisciplinary Digital Publishing Institute (MDPI)
2 publications, 40%
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1
2
3
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- We do not take into account publications that without a DOI.
- Statistics recalculated only for publications connected to researchers, organizations and labs registered on the platform.
- Statistics recalculated weekly.
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Uspenskaya A. A. et al. Influence of the dipeptide linker configuration on the activity of PSMA ligands // Mendeleev Communications. 2020. Vol. 30. No. 6. pp. 756-759.
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Uspenskaya A. A., Machulkin A. E., Nimenko E. A., Shafikov R. R., Petrov S. A., Skvortsov D. A., Beloglazkina E. K., Majouga A. G., Shafikov R. R., Petrov S. B., Skvortsov D., Beloglazkina E. K., Majouga A. G. Influence of the dipeptide linker configuration on the activity of PSMA ligands // Mendeleev Communications. 2020. Vol. 30. No. 6. pp. 756-759.
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TY - JOUR
DO - 10.1016/j.mencom.2020.11.022
UR - https://doi.org/10.1016%2Fj.mencom.2020.11.022
TI - Influence of the dipeptide linker configuration on the activity of PSMA ligands
T2 - Mendeleev Communications
AU - Uspenskaya, Anastasiya A
AU - Machulkin, Alexey E.
AU - Nimenko, Ekaterina A.
AU - Shafikov, Radik R
AU - Petrov, Stanislav A
AU - Skvortsov, Dmitry A.
AU - Beloglazkina, Elena K
AU - Majouga, Alexander G.
AU - Shafikov, Radik R
AU - Petrov, Stanislav B.
AU - Skvortsov, Dmitry
AU - Beloglazkina, Elena K.
AU - Majouga, Alexander G.
PY - 2020
DA - 2020/11/01 00:00:00
PB - Elsevier
SP - 756-759
IS - 6
VL - 30
SN - 0959-9436
SN - 1364-551X
ER -
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@article{2020_Uspenskaya,
author = {Anastasiya A Uspenskaya and Alexey E. Machulkin and Ekaterina A. Nimenko and Radik R Shafikov and Stanislav A Petrov and Dmitry A. Skvortsov and Elena K Beloglazkina and Alexander G. Majouga and Radik R Shafikov and Stanislav B. Petrov and Dmitry Skvortsov and Elena K. Beloglazkina and Alexander G. Majouga},
title = {Influence of the dipeptide linker configuration on the activity of PSMA ligands},
journal = {Mendeleev Communications},
year = {2020},
volume = {30},
publisher = {Elsevier},
month = {nov},
url = {https://doi.org/10.1016%2Fj.mencom.2020.11.022},
number = {6},
pages = {756--759},
doi = {10.1016/j.mencom.2020.11.022}
}
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Uspenskaya, Anastasiya A., et al. āInfluence of the dipeptide linker configuration on the activity of PSMA ligands.ā Mendeleev Communications, vol. 30, no. 6, Nov. 2020, pp. 756-759. https://doi.org/10.1016%2Fj.mencom.2020.11.022.