том 51 издание 9 страницы 1298-1302

Synthetic studies on nemorosone via enantioselective intramolecular cyclopropanation

Тип публикацииJournal Article
Дата публикации2010-03-01
scimago Q3
wos Q3
БС2
SJR0.334
CiteScore3.2
Impact factor1.5
ISSN00404039, 18733581
Organic Chemistry
Drug Discovery
Biochemistry
Краткое описание
This Letter describes synthetic studies of nemorosone via enantioselective intramolecular cyclopropanation. For the total synthesis of nemorosone, three potential intermediates were evaluated through the efficiency of three sequential reactions, namely, their intramolecular cyclopropanation, dimethylation of the resultant cyclopropanes, and ring-opening reaction of the alkylated cyclopropanes. As a result, α-diazomethyl ketone 10c was found to be the most suitable. The enantioselective intramolecular cyclopropanation to construct the bicyclo[3.3.1]nonane core and preparation of the compound with all the correct stereogenic centers of nemorosone are also described.
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ГОСТ |
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Abe M., Saito A., NAKADA M. Synthetic studies on nemorosone via enantioselective intramolecular cyclopropanation // Tetrahedron Letters. 2010. Vol. 51. No. 9. pp. 1298-1302.
ГОСТ со всеми авторами (до 50) Скопировать
Abe M., Saito A., NAKADA M. Synthetic studies on nemorosone via enantioselective intramolecular cyclopropanation // Tetrahedron Letters. 2010. Vol. 51. No. 9. pp. 1298-1302.
RIS |
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TY - JOUR
DO - 10.1016/j.tetlet.2009.12.147
UR - https://doi.org/10.1016/j.tetlet.2009.12.147
TI - Synthetic studies on nemorosone via enantioselective intramolecular cyclopropanation
T2 - Tetrahedron Letters
AU - Abe, Masahito
AU - Saito, Aya
AU - NAKADA, Masahisa
PY - 2010
DA - 2010/03/01
PB - Elsevier
SP - 1298-1302
IS - 9
VL - 51
SN - 0040-4039
SN - 1873-3581
ER -
BibTex |
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BibTex (до 50 авторов) Скопировать
@article{2010_Abe,
author = {Masahito Abe and Aya Saito and Masahisa NAKADA},
title = {Synthetic studies on nemorosone via enantioselective intramolecular cyclopropanation},
journal = {Tetrahedron Letters},
year = {2010},
volume = {51},
publisher = {Elsevier},
month = {mar},
url = {https://doi.org/10.1016/j.tetlet.2009.12.147},
number = {9},
pages = {1298--1302},
doi = {10.1016/j.tetlet.2009.12.147}
}
MLA
Цитировать
Abe, Masahito, et al. “Synthetic studies on nemorosone via enantioselective intramolecular cyclopropanation.” Tetrahedron Letters, vol. 51, no. 9, Mar. 2010, pp. 1298-1302. https://doi.org/10.1016/j.tetlet.2009.12.147.