Convenient entry to N-pyridinylureas with pharmaceutically privileged oxadiazole substituents via the acid-catalyzed C H activation of N-oxides
Publication type: Journal Article
Publication date: 2019-10-01
scimago Q3
wos Q3
SJR: 0.334
CiteScore: 3.2
Impact factor: 1.5
ISSN: 00404039, 18733581
Organic Chemistry
Drug Discovery
Biochemistry
Abstract
Pyridine-N-oxides bearing a pharmacophoric oxadiazole moiety could be C H functionalized via the acid-catalyzed reaction with dialkylcyanamides, providing access to hitherto undescribed pyridine-2-yl substituted ureas, which have potential as “lead-like” scaffolds for medicinal chemistry. Atom-economy, environmental friendliness (no halide-containing or toxic reagents), simple work-up, as well as scalability are the main advantages of the employed procedure.
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Total citations:
21
Citations from 2024:
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(19%)
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GOST
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Geyl K. et al. Convenient entry to N-pyridinylureas with pharmaceutically privileged oxadiazole substituents via the acid-catalyzed C H activation of N-oxides // Tetrahedron Letters. 2019. Vol. 60. No. 40. p. 151108.
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Geyl K., Matveevskaya V. V., Zelenkov L. E., Tarasenko M., Boyarskiy V. P. Convenient entry to N-pyridinylureas with pharmaceutically privileged oxadiazole substituents via the acid-catalyzed C H activation of N-oxides // Tetrahedron Letters. 2019. Vol. 60. No. 40. p. 151108.
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RIS
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TY - JOUR
DO - 10.1016/j.tetlet.2019.151108
UR - https://doi.org/10.1016/j.tetlet.2019.151108
TI - Convenient entry to N-pyridinylureas with pharmaceutically privileged oxadiazole substituents via the acid-catalyzed C H activation of N-oxides
T2 - Tetrahedron Letters
AU - Geyl, Kirill
AU - Matveevskaya, Vladislava V
AU - Zelenkov, Lev E
AU - Tarasenko, Marina
AU - Boyarskiy, Vadim P
PY - 2019
DA - 2019/10/01
PB - Elsevier
SP - 151108
IS - 40
VL - 60
SN - 0040-4039
SN - 1873-3581
ER -
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BibTex (up to 50 authors)
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@article{2019_Geyl,
author = {Kirill Geyl and Vladislava V Matveevskaya and Lev E Zelenkov and Marina Tarasenko and Vadim P Boyarskiy},
title = {Convenient entry to N-pyridinylureas with pharmaceutically privileged oxadiazole substituents via the acid-catalyzed C H activation of N-oxides},
journal = {Tetrahedron Letters},
year = {2019},
volume = {60},
publisher = {Elsevier},
month = {oct},
url = {https://doi.org/10.1016/j.tetlet.2019.151108},
number = {40},
pages = {151108},
doi = {10.1016/j.tetlet.2019.151108}
}
Cite this
MLA
Copy
Geyl, Kirill, et al. “Convenient entry to N-pyridinylureas with pharmaceutically privileged oxadiazole substituents via the acid-catalyzed C H activation of N-oxides.” Tetrahedron Letters, vol. 60, no. 40, Oct. 2019, p. 151108. https://doi.org/10.1016/j.tetlet.2019.151108.