Synthesis and biological activity of peptide antagonists of luliberin (luteinizing hormone-releasing hormone)
Publication type: Journal Article
Publication date: 1979-08-01
scimago Q1
wos Q1
SJR: 1.801
CiteScore: 11.5
Impact factor: 6.8
ISSN: 00222623, 15204804
PubMed ID:
385877
Drug Discovery
Molecular Medicine
Abstract
A series of des-His2 octa- and nonapeptide analogues of luliberin (luteinizing hormone-releasing hormone) with modifications in the 1 and 6 positions, and in some instances the 10 position, has been prepared. Some of these analogues are potent inhibitors of luliberin in vitro and in vivo. The use of ultraviolet absorption measurements for evaluating peptides containing tyrosine and tryptophan is described. An efficient synthesis of O-methyl-d-tyrosine is reported.
Found
Nothing found, try to update filter.
Top-30
Journals
|
1
2
|
|
|
Chemistry of Natural Compounds
2 publications, 10%
|
|
|
Contraception
2 publications, 10%
|
|
|
International journal of peptide & protein research
2 publications, 10%
|
|
|
Journal of Medicinal Chemistry
1 publication, 5%
|
|
|
Journal of the American Chemical Society
1 publication, 5%
|
|
|
Journal of Organic Chemistry
1 publication, 5%
|
|
|
Tetrahedron Asymmetry
1 publication, 5%
|
|
|
Chromatographia
1 publication, 5%
|
|
|
Molecular Aspects of Medicine
1 publication, 5%
|
|
|
Peptides
1 publication, 5%
|
|
|
Tetrahedron Letters
1 publication, 5%
|
|
|
Chemischer Informationsdienst
1 publication, 5%
|
|
|
Journal für praktische Chemie
1 publication, 5%
|
|
|
Organic Preparations and Procedures International
1 publication, 5%
|
|
|
Topics in Heterocyclic Chemistry
1 publication, 5%
|
|
|
Synthesis
1 publication, 5%
|
|
|
1
2
|
Publishers
|
1
2
3
4
5
6
|
|
|
Elsevier
6 publications, 30%
|
|
|
Springer Nature
4 publications, 20%
|
|
|
Wiley
4 publications, 20%
|
|
|
American Chemical Society (ACS)
3 publications, 15%
|
|
|
Taylor & Francis
1 publication, 5%
|
|
|
Georg Thieme Verlag KG
1 publication, 5%
|
|
|
1
2
3
4
5
6
|
- We do not take into account publications without a DOI.
- Statistics recalculated weekly.
Are you a researcher?
Create a profile to get free access to personal recommendations for colleagues and new articles.
Metrics
20
Total citations:
20
Citations from 2024:
0
Cite this
GOST |
RIS |
BibTex |
MLA
Cite this
GOST
Copy
Moersch G. W. et al. Synthesis and biological activity of peptide antagonists of luliberin (luteinizing hormone-releasing hormone) // Journal of Medicinal Chemistry. 1979. Vol. 22. No. 8. pp. 935-943.
GOST all authors (up to 50)
Copy
Moersch G. W., Rebstock M. C., Wittle E. L., Tinney F. J., Nicolaides E. D., Hutt M. P., Mich T. F., Vandenbelt J. M., Edgren R. E. Synthesis and biological activity of peptide antagonists of luliberin (luteinizing hormone-releasing hormone) // Journal of Medicinal Chemistry. 1979. Vol. 22. No. 8. pp. 935-943.
Cite this
RIS
Copy
TY - JOUR
DO - 10.1021/jm00194a010
UR - https://doi.org/10.1021/jm00194a010
TI - Synthesis and biological activity of peptide antagonists of luliberin (luteinizing hormone-releasing hormone)
T2 - Journal of Medicinal Chemistry
AU - Moersch, G. W.
AU - Rebstock, M C
AU - Wittle, E L
AU - Tinney, F J
AU - Nicolaides, E D
AU - Hutt, M. P.
AU - Mich, T F
AU - Vandenbelt, J M
AU - Edgren, R E
PY - 1979
DA - 1979/08/01
PB - American Chemical Society (ACS)
SP - 935-943
IS - 8
VL - 22
PMID - 385877
SN - 0022-2623
SN - 1520-4804
ER -
Cite this
BibTex (up to 50 authors)
Copy
@article{1979_Moersch,
author = {G. W. Moersch and M C Rebstock and E L Wittle and F J Tinney and E D Nicolaides and M. P. Hutt and T F Mich and J M Vandenbelt and R E Edgren},
title = {Synthesis and biological activity of peptide antagonists of luliberin (luteinizing hormone-releasing hormone)},
journal = {Journal of Medicinal Chemistry},
year = {1979},
volume = {22},
publisher = {American Chemical Society (ACS)},
month = {aug},
url = {https://doi.org/10.1021/jm00194a010},
number = {8},
pages = {935--943},
doi = {10.1021/jm00194a010}
}
Cite this
MLA
Copy
Moersch, G. W., et al. “Synthesis and biological activity of peptide antagonists of luliberin (luteinizing hormone-releasing hormone).” Journal of Medicinal Chemistry, vol. 22, no. 8, Aug. 1979, pp. 935-943. https://doi.org/10.1021/jm00194a010.