том 18 издание 7 страницы 3740-3746

Polymorphism of Sildenafil: A New Metastable Desolvate

Тип публикацииJournal Article
Дата публикации2018-06-12
scimago Q2
wos Q1
БС1
SJR0.633
CiteScore5.6
Impact factor3.4
ISSN15287483, 15287505
General Chemistry
Condensed Matter Physics
General Materials Science
Краткое описание
A new anhydrous polymorph of the free base of sildenafil and two solvates (acetonitrile and propanenitrile) have been discovered and fully characterized. The new polymorph can be considered a desolvate of the acetonitrile solvate and is related to the most stable form I by morphotropism. The new polymorph can only be obtained by desolvation of the acetonitrile solvate. Thus, this study is a new example of the importance of this multicomponent family of solid forms in the discovery of new polymorphs of active pharmaceutical ingredients.
Найдено 
Найдено 

Топ-30

Журналы

1
2
3
4
5
6
CrystEngComm
6 публикаций, 26.09%
Crystal Growth and Design
3 публикации, 13.04%
Crystals
1 публикация, 4.35%
Pharmaceuticals
1 публикация, 4.35%
Journal of Solution Chemistry
1 публикация, 4.35%
Journal of Pharmaceutical Sciences
1 публикация, 4.35%
Acta Crystallographica Section B: Structural Science, Crystal Engineering and Materials
1 публикация, 4.35%
Journal of Chemical Information and Modeling
1 публикация, 4.35%
Zeitschrift fur Naturforschung - Section B Journal of Chemical Sciences
1 публикация, 4.35%
Zeitschrift fur Physikalische Chemie
1 публикация, 4.35%
Journal of Molecular Liquids
1 публикация, 4.35%
Journal of Pharmaceutical and Biomedical Analysis Open
1 публикация, 4.35%
IUCrJ
1 публикация, 4.35%
International Journal of Pharmaceutics
1 публикация, 4.35%
1
2
3
4
5
6

Издатели

1
2
3
4
5
6
Royal Society of Chemistry (RSC)
6 публикаций, 26.09%
Elsevier
5 публикаций, 21.74%
American Chemical Society (ACS)
4 публикации, 17.39%
MDPI
2 публикации, 8.7%
International Union of Crystallography (IUCr)
2 публикации, 8.7%
Walter de Gruyter
2 публикации, 8.7%
Springer Nature
1 публикация, 4.35%
IntechOpen
1 публикация, 4.35%
1
2
3
4
5
6
  • Мы не учитываем публикации, у которых нет DOI.
  • Статистика публикаций обновляется еженедельно.

Вы ученый?

Создайте профиль, чтобы получать персональные рекомендации коллег, конференций и новых статей.
Метрики
23
Поделиться
Цитировать
ГОСТ |
Цитировать
Barbas R., Font-Bardia M., Prohens R. Polymorphism of Sildenafil: A New Metastable Desolvate // Crystal Growth and Design. 2018. Vol. 18. No. 7. pp. 3740-3746.
ГОСТ со всеми авторами (до 50) Скопировать
Barbas R., Font-Bardia M., Prohens R. Polymorphism of Sildenafil: A New Metastable Desolvate // Crystal Growth and Design. 2018. Vol. 18. No. 7. pp. 3740-3746.
RIS |
Цитировать
TY - JOUR
DO - 10.1021/acs.cgd.8b00683
UR - https://doi.org/10.1021/acs.cgd.8b00683
TI - Polymorphism of Sildenafil: A New Metastable Desolvate
T2 - Crystal Growth and Design
AU - Barbas, Rafael
AU - Font-Bardia, M.
AU - Prohens, Rafel
PY - 2018
DA - 2018/06/12
PB - American Chemical Society (ACS)
SP - 3740-3746
IS - 7
VL - 18
SN - 1528-7483
SN - 1528-7505
ER -
BibTex |
Цитировать
BibTex (до 50 авторов) Скопировать
@article{2018_Barbas,
author = {Rafael Barbas and M. Font-Bardia and Rafel Prohens},
title = {Polymorphism of Sildenafil: A New Metastable Desolvate},
journal = {Crystal Growth and Design},
year = {2018},
volume = {18},
publisher = {American Chemical Society (ACS)},
month = {jun},
url = {https://doi.org/10.1021/acs.cgd.8b00683},
number = {7},
pages = {3740--3746},
doi = {10.1021/acs.cgd.8b00683}
}
MLA
Цитировать
Barbas, Rafael, et al. “Polymorphism of Sildenafil: A New Metastable Desolvate.” Crystal Growth and Design, vol. 18, no. 7, Jun. 2018, pp. 3740-3746. https://doi.org/10.1021/acs.cgd.8b00683.