volume 20 issue 4 pages 1130-1133

Copper-Mediated Reactions of Nitriles with Nitromethanes: Aza-Henry Reactions and Nitrile Hydrations

Publication typeJournal Article
Publication date2018-02-07
scimago Q1
wos Q1
SJR1.235
CiteScore8.7
Impact factor5.0
ISSN15237060, 15237052
Organic Chemistry
Biochemistry
Physical and Theoretical Chemistry
Abstract
In this study, the first aza-Henry reaction of nitriles with nitromethane in a CuI/Cs2CO3/DBU system is described. The process was conveniently and directly used for the synthesis of β-aminonitroalkenes 2a-x and tolerated aryl-, alkyl-, hetaryl-, alkenyl-, and alkynylnitriles. The resulting aminonitroalkenes 2 could be successfully transformed to the corresponding 2-nitroacetophenones, 2-amino-1-halonitroalkenes, 2-alkylaminonitroalkenes, or 3-nitropyridines. In the presence of H2O, the aza-Henry reaction turned the reaction path to the nitrile hydration to exclusively yield the amides 3a-s.
Found 
Found 

Top-30

Journals

1
2
Tetrahedron
2 publications, 13.33%
Organic and Biomolecular Chemistry
2 publications, 13.33%
Russian Chemical Reviews
2 publications, 13.33%
Journal of Organic Chemistry
1 publication, 6.67%
ChemCatChem
1 publication, 6.67%
Organic Letters
1 publication, 6.67%
Chemical Communications
1 publication, 6.67%
Journal of Biomolecular Structure and Dynamics
1 publication, 6.67%
Synlett
1 publication, 6.67%
Journal of the American Chemical Society
1 publication, 6.67%
Russian Journal of Organic Chemistry
1 publication, 6.67%
1
2

Publishers

1
2
3
American Chemical Society (ACS)
3 publications, 20%
Royal Society of Chemistry (RSC)
3 publications, 20%
Elsevier
2 publications, 13.33%
Wiley
2 publications, 13.33%
Autonomous Non-profit Organization Editorial Board of the journal Uspekhi Khimii
2 publications, 13.33%
Taylor & Francis
1 publication, 6.67%
Georg Thieme Verlag KG
1 publication, 6.67%
Pleiades Publishing
1 publication, 6.67%
1
2
3
  • We do not take into account publications without a DOI.
  • Statistics recalculated weekly.

Are you a researcher?

Create a profile to get free access to personal recommendations for colleagues and new articles.
Metrics
15
Share
Cite this
GOST |
Cite this
GOST Copy
Kuwabara J., Sawada Y., Yoshimatsu M. Copper-Mediated Reactions of Nitriles with Nitromethanes: Aza-Henry Reactions and Nitrile Hydrations // Organic Letters. 2018. Vol. 20. No. 4. pp. 1130-1133.
GOST all authors (up to 50) Copy
Kuwabara J., Sawada Y., Yoshimatsu M. Copper-Mediated Reactions of Nitriles with Nitromethanes: Aza-Henry Reactions and Nitrile Hydrations // Organic Letters. 2018. Vol. 20. No. 4. pp. 1130-1133.
RIS |
Cite this
RIS Copy
TY - JOUR
DO - 10.1021/acs.orglett.8b00058
UR - https://doi.org/10.1021/acs.orglett.8b00058
TI - Copper-Mediated Reactions of Nitriles with Nitromethanes: Aza-Henry Reactions and Nitrile Hydrations
T2 - Organic Letters
AU - Kuwabara, Jun
AU - Sawada, Yoshiharu
AU - Yoshimatsu, Mitsuhiro
PY - 2018
DA - 2018/02/07
PB - American Chemical Society (ACS)
SP - 1130-1133
IS - 4
VL - 20
PMID - 29412678
SN - 1523-7060
SN - 1523-7052
ER -
BibTex |
Cite this
BibTex (up to 50 authors) Copy
@article{2018_Kuwabara,
author = {Jun Kuwabara and Yoshiharu Sawada and Mitsuhiro Yoshimatsu},
title = {Copper-Mediated Reactions of Nitriles with Nitromethanes: Aza-Henry Reactions and Nitrile Hydrations},
journal = {Organic Letters},
year = {2018},
volume = {20},
publisher = {American Chemical Society (ACS)},
month = {feb},
url = {https://doi.org/10.1021/acs.orglett.8b00058},
number = {4},
pages = {1130--1133},
doi = {10.1021/acs.orglett.8b00058}
}
MLA
Cite this
MLA Copy
Kuwabara, Jun, et al. “Copper-Mediated Reactions of Nitriles with Nitromethanes: Aza-Henry Reactions and Nitrile Hydrations.” Organic Letters, vol. 20, no. 4, Feb. 2018, pp. 1130-1133. https://doi.org/10.1021/acs.orglett.8b00058.