том 21 издание 5 страницы 1426-1429

Synthesis of β-Arylethenesulfonyl Fluoride via Pd-Catalyzed Nondirected C-H Alkenylation.

Тип публикацииJournal Article
Дата публикации2019-02-20
SCImago Q1
Tоп 10% SCImago
WOS Q1
БС1
SJR1.007
CiteScore7.7
Impact factor4.7
ISSN15237060, 15237052
Organic Chemistry
Biochemistry
Physical and Theoretical Chemistry
Краткое описание
A rapid synthesis of β-arylethenesulfonyl fluorides is realized using ligand-accelerated Pd(II)-catalyzed nondirected C-H alkenylation of simple arenes. The newly developed electron-deficient 2-pyridone ligand is crucial for this transformation with arenes as limiting reagent. This protocol features a broad substrate scope and good functional group tolerance. Late-stage functionalization of various pharmaceuticals and their further click manipulations demonstrate this procedure to be highly valuable.
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ГОСТ |
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Chen X. et al. Synthesis of β-Arylethenesulfonyl Fluoride via Pd-Catalyzed Nondirected C-H Alkenylation. // Organic Letters. 2019. Vol. 21. No. 5. pp. 1426-1429.
ГОСТ со всеми авторами (до 50) Скопировать
Chen X., Wu Y., Zhou J., Wang P., Yu J. Synthesis of β-Arylethenesulfonyl Fluoride via Pd-Catalyzed Nondirected C-H Alkenylation. // Organic Letters. 2019. Vol. 21. No. 5. pp. 1426-1429.
RIS |
Цитировать
TY - JOUR
DO - 10.1021/acs.orglett.9b00165
UR - https://doi.org/10.1021/acs.orglett.9b00165
TI - Synthesis of β-Arylethenesulfonyl Fluoride via Pd-Catalyzed Nondirected C-H Alkenylation.
T2 - Organic Letters
AU - Chen, Xiao-Yue
AU - Wu, Yichen
AU - Zhou, Jian
AU - Wang, Peng
AU - Yu, Jinquan
PY - 2019
DA - 2019/02/20
PB - American Chemical Society (ACS)
SP - 1426-1429
IS - 5
VL - 21
PMID - 30785296
SN - 1523-7060
SN - 1523-7052
ER -
BibTex |
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BibTex (до 50 авторов) Скопировать
@article{2019_Chen,
author = {Xiao-Yue Chen and Yichen Wu and Jian Zhou and Peng Wang and Jinquan Yu},
title = {Synthesis of β-Arylethenesulfonyl Fluoride via Pd-Catalyzed Nondirected C-H Alkenylation.},
journal = {Organic Letters},
year = {2019},
volume = {21},
publisher = {American Chemical Society (ACS)},
month = {feb},
url = {https://doi.org/10.1021/acs.orglett.9b00165},
number = {5},
pages = {1426--1429},
doi = {10.1021/acs.orglett.9b00165}
}
MLA
Цитировать
Chen, Xiao-Yue, et al. “Synthesis of β-Arylethenesulfonyl Fluoride via Pd-Catalyzed Nondirected C-H Alkenylation..” Organic Letters, vol. 21, no. 5, Feb. 2019, pp. 1426-1429. https://doi.org/10.1021/acs.orglett.9b00165.
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