том 134 издание 23 страницы 9721-9726

Directed Metal (Oxo) Aliphatic C–H Hydroxylations: Overriding Substrate Bias

Тип публикацииJournal Article
Дата публикации2012-06-01
SCImago Q1
Tоп 10% SCImago
WOS Q1
БС1
SJR5.491
CiteScore22
Impact factor16.6
ISSN00027863, 15205126
General Chemistry
Catalysis
Biochemistry
Colloid and Surface Chemistry
Краткое описание
The first general strategy for a directing effect on metal (oxo)-promoted C-H hydroxylations is described. Carboxylic acid moieties on the substrate overcome unfavorable electronic, steric, and stereoelectronic biases in C-H hydroxylations catalyzed by the non-heme iron complex Fe(PDP). In a demonstration of the power of this directing effect, C-H oxidation is diverted away from an electronically favored C-1 H abstraction/rearrangement pathway in the paclitaxel framework to enable installation of C-2 oxidation in the naturally occurring oxidation state and stereoconfiguration.
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ГОСТ |
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Bigi M. A., Reed S. A., White M. Directed Metal (Oxo) Aliphatic C–H Hydroxylations: Overriding Substrate Bias // Journal of the American Chemical Society. 2012. Vol. 134. No. 23. pp. 9721-9726.
ГОСТ со всеми авторами (до 50) Скопировать
Bigi M. A., Reed S. A., White M. Directed Metal (Oxo) Aliphatic C–H Hydroxylations: Overriding Substrate Bias // Journal of the American Chemical Society. 2012. Vol. 134. No. 23. pp. 9721-9726.
RIS |
Цитировать
TY - JOUR
DO - 10.1021/ja301685r
UR - https://doi.org/10.1021/ja301685r
TI - Directed Metal (Oxo) Aliphatic C–H Hydroxylations: Overriding Substrate Bias
T2 - Journal of the American Chemical Society
AU - Bigi, Marinus A
AU - Reed, Sean A
AU - White, M.
PY - 2012
DA - 2012/06/01
PB - American Chemical Society (ACS)
SP - 9721-9726
IS - 23
VL - 134
PMID - 22607637
SN - 0002-7863
SN - 1520-5126
ER -
BibTex |
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BibTex (до 50 авторов) Скопировать
@article{2012_Bigi,
author = {Marinus A Bigi and Sean A Reed and M. White},
title = {Directed Metal (Oxo) Aliphatic C–H Hydroxylations: Overriding Substrate Bias},
journal = {Journal of the American Chemical Society},
year = {2012},
volume = {134},
publisher = {American Chemical Society (ACS)},
month = {jun},
url = {https://doi.org/10.1021/ja301685r},
number = {23},
pages = {9721--9726},
doi = {10.1021/ja301685r}
}
MLA
Цитировать
Bigi, Marinus A., et al. “Directed Metal (Oxo) Aliphatic C–H Hydroxylations: Overriding Substrate Bias.” Journal of the American Chemical Society, vol. 134, no. 23, Jun. 2012, pp. 9721-9726. https://doi.org/10.1021/ja301685r.
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