Discovery and Optimization of a Novel Series of Thrombin Receptor (PAR-1) Antagonists: Potent, Selective Peptide Mimetics Based on Indole and Indazole Templates
Han-Cheng Zhang
1
,
Claudia K. Derian
1
,
Patricia Andrade-Gordon
1
,
William J. Hoekstra
1
,
David F. McComsey
1
,
Kimberly B. White
1
,
Brenda L. Poulter
1
,
Michael F. Addo
1
,
Wai-man Cheung
1
,
Bruce P. Damiano
1
,
Donna Oksenberg
1
,
Elwood E. Reynolds
1
,
Anjali Pandey
1
,
Robert M. Scarborough
1
,
Bruce E Maryanoff
1
1
Drug Discovery, The R. W. Johnson Pharmaceutical Research Institute, Spring House, Pennsylvania 19477, and COR Therapeutics, Inc., South San Francisco, California 94080
|
Publication type: Journal Article
Publication date: 2001-03-01
scimago Q1
wos Q1
SJR: 1.801
CiteScore: 11.5
Impact factor: 6.8
ISSN: 00222623, 15204804
PubMed ID:
11297447
Drug Discovery
Molecular Medicine
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69
Total citations:
69
Citations from 2024:
2
(2.9%)
Cite this
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MLA
Cite this
GOST
Copy
Zhang H. et al. Discovery and Optimization of a Novel Series of Thrombin Receptor (PAR-1) Antagonists: Potent, Selective Peptide Mimetics Based on Indole and Indazole Templates // Journal of Medicinal Chemistry. 2001. Vol. 44. No. 7. pp. 1021-1024.
GOST all authors (up to 50)
Copy
Zhang H., Derian C. K., Andrade-Gordon P., Hoekstra W. J., McComsey D. F., White K. B., Poulter B. L., Addo M. F., Cheung W., Damiano B. P., Oksenberg D., Reynolds E. E., Pandey A., Scarborough R. M., Maryanoff B. E. Discovery and Optimization of a Novel Series of Thrombin Receptor (PAR-1) Antagonists: Potent, Selective Peptide Mimetics Based on Indole and Indazole Templates // Journal of Medicinal Chemistry. 2001. Vol. 44. No. 7. pp. 1021-1024.
Cite this
RIS
Copy
TY - JOUR
DO - 10.1021/jm000506s
UR - https://doi.org/10.1021/jm000506s
TI - Discovery and Optimization of a Novel Series of Thrombin Receptor (PAR-1) Antagonists: Potent, Selective Peptide Mimetics Based on Indole and Indazole Templates
T2 - Journal of Medicinal Chemistry
AU - Zhang, Han-Cheng
AU - Derian, Claudia K.
AU - Andrade-Gordon, Patricia
AU - Hoekstra, William J.
AU - McComsey, David F.
AU - White, Kimberly B.
AU - Poulter, Brenda L.
AU - Addo, Michael F.
AU - Cheung, Wai-man
AU - Damiano, Bruce P.
AU - Oksenberg, Donna
AU - Reynolds, Elwood E.
AU - Pandey, Anjali
AU - Scarborough, Robert M.
AU - Maryanoff, Bruce E
PY - 2001
DA - 2001/03/01
PB - American Chemical Society (ACS)
SP - 1021-1024
IS - 7
VL - 44
PMID - 11297447
SN - 0022-2623
SN - 1520-4804
ER -
Cite this
BibTex (up to 50 authors)
Copy
@article{2001_Zhang,
author = {Han-Cheng Zhang and Claudia K. Derian and Patricia Andrade-Gordon and William J. Hoekstra and David F. McComsey and Kimberly B. White and Brenda L. Poulter and Michael F. Addo and Wai-man Cheung and Bruce P. Damiano and Donna Oksenberg and Elwood E. Reynolds and Anjali Pandey and Robert M. Scarborough and Bruce E Maryanoff},
title = {Discovery and Optimization of a Novel Series of Thrombin Receptor (PAR-1) Antagonists: Potent, Selective Peptide Mimetics Based on Indole and Indazole Templates},
journal = {Journal of Medicinal Chemistry},
year = {2001},
volume = {44},
publisher = {American Chemical Society (ACS)},
month = {mar},
url = {https://doi.org/10.1021/jm000506s},
number = {7},
pages = {1021--1024},
doi = {10.1021/jm000506s}
}
Cite this
MLA
Copy
Zhang, Han-Cheng, et al. “Discovery and Optimization of a Novel Series of Thrombin Receptor (PAR-1) Antagonists: Potent, Selective Peptide Mimetics Based on Indole and Indazole Templates.” Journal of Medicinal Chemistry, vol. 44, no. 7, Mar. 2001, pp. 1021-1024. https://doi.org/10.1021/jm000506s.