Studies on cardiovascular agents. 6. Synthesis and coronary vasodilating and antihypertensive activities of 1,2,4-triazolo[1,5-a]pyrimidines fused to heterocyclic systems
Тип публикации: Journal Article
Дата публикации: 1980-08-01
SCImago Q1
Tоп 10% SCImago
WOS Q1
БС1
SJR: 1.726
CiteScore: 11.1
Impact factor: 7.3
ISSN: 00222623, 15204804
PubMed ID:
7401118
Drug Discovery
Molecular Medicine
Краткое описание
The synthesis and coronary vasodilating and antihypertensive activities of 1,2,4-triazolo[1,5-a]pyrimidines fused to pyrrole, thiophene, pyran, pyridine, and pyridazine are described. Among these compounds, 8-tert-butyl-7,8-dihydro-5-methyl-6H-pyrrolo[3,2-e][1,2,4]triazolo[1,5-a]pyrimidine (23) was found to be the most promising potential cardiovascular agent, having been shown to be more potent in coronary vasodilating activity than trapidil [7-diethylamino)-5-methyl-1,2,4-triazolo[1,5-a]pyrimidine] and approximately equipotent to guanethidine sulfate in antihypertensive activity.
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52
Всего цитирований:
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ГОСТ
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Sato Y. et al. Studies on cardiovascular agents. 6. Synthesis and coronary vasodilating and antihypertensive activities of 1,2,4-triazolo[1,5-a]pyrimidines fused to heterocyclic systems // Journal of Medicinal Chemistry. 1980. Vol. 23. No. 8. pp. 927-937.
ГОСТ со всеми авторами (до 50)
Скопировать
Sato Y., SHIMOJI Y., FUJITA H., NISHINO H., Mizuno H., Kobayashi S., Kumakura S. Studies on cardiovascular agents. 6. Synthesis and coronary vasodilating and antihypertensive activities of 1,2,4-triazolo[1,5-a]pyrimidines fused to heterocyclic systems // Journal of Medicinal Chemistry. 1980. Vol. 23. No. 8. pp. 927-937.
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RIS
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TY - JOUR
DO - 10.1021/jm00182a021
UR - https://doi.org/10.1021/jm00182a021
TI - Studies on cardiovascular agents. 6. Synthesis and coronary vasodilating and antihypertensive activities of 1,2,4-triazolo[1,5-a]pyrimidines fused to heterocyclic systems
T2 - Journal of Medicinal Chemistry
AU - Sato, Yasunobu
AU - SHIMOJI, Yasuo
AU - FUJITA, HIROSHI
AU - NISHINO, Hiroshi
AU - Mizuno, Hiroshi
AU - Kobayashi, Shinsaku
AU - Kumakura, Seiji
PY - 1980
DA - 1980/08/01
PB - American Chemical Society (ACS)
SP - 927-937
IS - 8
VL - 23
PMID - 7401118
SN - 0022-2623
SN - 1520-4804
ER -
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BibTex (до 50 авторов)
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@article{1980_Sato,
author = {Yasunobu Sato and Yasuo SHIMOJI and HIROSHI FUJITA and Hiroshi NISHINO and Hiroshi Mizuno and Shinsaku Kobayashi and Seiji Kumakura},
title = {Studies on cardiovascular agents. 6. Synthesis and coronary vasodilating and antihypertensive activities of 1,2,4-triazolo[1,5-a]pyrimidines fused to heterocyclic systems},
journal = {Journal of Medicinal Chemistry},
year = {1980},
volume = {23},
publisher = {American Chemical Society (ACS)},
month = {aug},
url = {https://doi.org/10.1021/jm00182a021},
number = {8},
pages = {927--937},
doi = {10.1021/jm00182a021}
}
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MLA
Скопировать
Sato, Yasunobu, et al. “Studies on cardiovascular agents. 6. Synthesis and coronary vasodilating and antihypertensive activities of 1,2,4-triazolo[1,5-a]pyrimidines fused to heterocyclic systems.” Journal of Medicinal Chemistry, vol. 23, no. 8, Aug. 1980, pp. 927-937. https://doi.org/10.1021/jm00182a021.
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