том 2 издание 13 страницы 1827-1830

Synthesis of Partially Modified Retro and Retroinverso ψ[NHCH(CF3)]-Peptides

Тип публикацииJournal Article
Дата публикации2000-05-27
scimago Q1
wos Q1
БС1
SJR1.235
CiteScore8.7
Impact factor5
ISSN15237060, 15237052
Organic Chemistry
Biochemistry
Physical and Theoretical Chemistry
Краткое описание
[reaction: see text] Asymmetric conjugate additions of chiral alpha-amino esters to chiral 4-CF(3) Michael-acceptors were exploited to prepare a small library of enantiomerically pure partially modified retropeptides having a psi[NHCH(CF(3))] unit as a possible mimic of the classical psi(NHCO) retropeptide unit. Yields were nearly quantitative, and the stereoselectivity, which is controlled mainly by the nitrogen nucleophile, was progressively higher with increasing the steric bulk of the alpha-amino ester side-chain R(1).
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ГОСТ |
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Volonterio A., Bravo P., Zanda M. Synthesis of Partially Modified Retro and Retroinverso ψ[NHCH(CF3)]-Peptides // Organic Letters. 2000. Vol. 2. No. 13. pp. 1827-1830.
ГОСТ со всеми авторами (до 50) Скопировать
Volonterio A., Bravo P., Zanda M. Synthesis of Partially Modified Retro and Retroinverso ψ[NHCH(CF3)]-Peptides // Organic Letters. 2000. Vol. 2. No. 13. pp. 1827-1830.
RIS |
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TY - JOUR
DO - 10.1021/ol005876p
UR - https://pubs.acs.org/doi/10.1021/ol005876p
TI - Synthesis of Partially Modified Retro and Retroinverso ψ[NHCH(CF3)]-Peptides
T2 - Organic Letters
AU - Volonterio, A.
AU - Bravo, Pierfrancesco
AU - Zanda, M.
PY - 2000
DA - 2000/05/27
PB - American Chemical Society (ACS)
SP - 1827-1830
IS - 13
VL - 2
PMID - 10891168
SN - 1523-7060
SN - 1523-7052
ER -
BibTex |
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BibTex (до 50 авторов) Скопировать
@article{2000_Volonterio,
author = {A. Volonterio and Pierfrancesco Bravo and M. Zanda},
title = {Synthesis of Partially Modified Retro and Retroinverso ψ[NHCH(CF3)]-Peptides},
journal = {Organic Letters},
year = {2000},
volume = {2},
publisher = {American Chemical Society (ACS)},
month = {may},
url = {https://pubs.acs.org/doi/10.1021/ol005876p},
number = {13},
pages = {1827--1830},
doi = {10.1021/ol005876p}
}
MLA
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Volonterio, A., et al. “Synthesis of Partially Modified Retro and Retroinverso ψ[NHCH(CF3)]-Peptides.” Organic Letters, vol. 2, no. 13, May. 2000, pp. 1827-1830. https://pubs.acs.org/doi/10.1021/ol005876p.