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A new facile synthesis of 3-amidoindole derivatives and their evaluation as potential GSK-3β inhibitors

Тип публикацииJournal Article
Дата публикации2010-01-14
scimago Q2
wos Q2
БС1
SJR0.600
CiteScore5.2
Impact factor2.7
ISSN14770520, 14770539
Organic Chemistry
Biochemistry
Physical and Theoretical Chemistry
Краткое описание
3-Amidoindoles were synthesized from commercially available arylhydrazines and propargylamines over Zn-salt mediated one pot procedure in excellent regioselectivity and up to 94% yield.
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ГОСТ |
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Pews-Davtyan A. et al. A new facile synthesis of 3-amidoindole derivatives and their evaluation as potential GSK-3β inhibitors // Organic and Biomolecular Chemistry. 2010. Vol. 8. No. 5. p. 1149.
ГОСТ со всеми авторами (до 50) Скопировать
Pews-Davtyan A., Tillack A., Schmöle A. C., Schmöle A., Ortinau S., Frech M. J., Rolfs A., Beller M. A new facile synthesis of 3-amidoindole derivatives and their evaluation as potential GSK-3β inhibitors // Organic and Biomolecular Chemistry. 2010. Vol. 8. No. 5. p. 1149.
RIS |
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TY - JOUR
DO - 10.1039/b920861e
UR - https://doi.org/10.1039/b920861e
TI - A new facile synthesis of 3-amidoindole derivatives and their evaluation as potential GSK-3β inhibitors
T2 - Organic and Biomolecular Chemistry
AU - Pews-Davtyan, Anahit
AU - Tillack, Annegret
AU - Schmöle, Anne Caroline
AU - Schmöle, Anne-Caroline
AU - Ortinau, Stefanie
AU - Frech, Moritz Johannes
AU - Rolfs, Arndt
AU - Beller, Matthias
PY - 2010
DA - 2010/01/14
PB - Royal Society of Chemistry (RSC)
SP - 1149
IS - 5
VL - 8
PMID - 20165807
SN - 1477-0520
SN - 1477-0539
ER -
BibTex |
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BibTex (до 50 авторов) Скопировать
@article{2010_Pews-Davtyan,
author = {Anahit Pews-Davtyan and Annegret Tillack and Anne Caroline Schmöle and Anne-Caroline Schmöle and Stefanie Ortinau and Moritz Johannes Frech and Arndt Rolfs and Matthias Beller},
title = {A new facile synthesis of 3-amidoindole derivatives and their evaluation as potential GSK-3β inhibitors},
journal = {Organic and Biomolecular Chemistry},
year = {2010},
volume = {8},
publisher = {Royal Society of Chemistry (RSC)},
month = {jan},
url = {https://doi.org/10.1039/b920861e},
number = {5},
pages = {1149},
doi = {10.1039/b920861e}
}
MLA
Цитировать
Pews-Davtyan, Anahit, et al. “A new facile synthesis of 3-amidoindole derivatives and their evaluation as potential GSK-3β inhibitors.” Organic and Biomolecular Chemistry, vol. 8, no. 5, Jan. 2010, p. 1149. https://doi.org/10.1039/b920861e.