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Convenient Synthesis of 2-Thioimidazolone/Menadione Conjugates via a Two-Step Sequence Starting with Direct Amination of Menadione
Publication type: Journal Article
Publication date: 2020-04-01
scimago Q2
wos Q3
SJR: 0.453
CiteScore: 3.6
Impact factor: 2.1
ISSN: 25099396
Catalysis
Organic Chemistry
Materials Science (miscellaneous)
Biomaterials
Abstract
A convenient route to conjugates of 2-thiohydantoins and menadione with linkers of various chemical nature through a two-stage reaction sequence (direct amination of the menadione with a functional amine followed by modification of a functional group) is presented. Optimal conditions for the direct amination of menadione using alkyl amines with substituents such as azide, alkyne, hydroxyl, amine, halogen, and carboxyl have been developed. Further modification of selected functionalities using CuAAC or esterification reactions with 2-thiohydantoines has been performed.
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Guk D. A. et al. Convenient Synthesis of 2-Thioimidazolone/Menadione Conjugates via a Two-Step Sequence Starting with Direct Amination of Menadione // SynOpen. 2020. Vol. 04. No. 02. pp. 38-43.
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Guk D. A. Convenient Synthesis of 2-Thioimidazolone/Menadione Conjugates via a Two-Step Sequence Starting with Direct Amination of Menadione // SynOpen. 2020. Vol. 04. No. 02. pp. 38-43.
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TY - JOUR
DO - 10.1055/s-0040-1707519
UR - http://www.thieme-connect.de/DOI/DOI?10.1055/s-0040-1707519
TI - Convenient Synthesis of 2-Thioimidazolone/Menadione Conjugates via a Two-Step Sequence Starting with Direct Amination of Menadione
T2 - SynOpen
AU - Guk, Dmitry A.
PY - 2020
DA - 2020/04/01
PB - Georg Thieme Verlag KG
SP - 38-43
IS - 02
VL - 04
SN - 2509-9396
ER -
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BibTex (up to 50 authors)
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@article{2020_Guk,
author = {Dmitry A. Guk},
title = {Convenient Synthesis of 2-Thioimidazolone/Menadione Conjugates via a Two-Step Sequence Starting with Direct Amination of Menadione},
journal = {SynOpen},
year = {2020},
volume = {04},
publisher = {Georg Thieme Verlag KG},
month = {apr},
url = {http://www.thieme-connect.de/DOI/DOI?10.1055/s-0040-1707519},
number = {02},
pages = {38--43},
doi = {10.1055/s-0040-1707519}
}
Cite this
MLA
Copy
Guk, Dmitry A., et al. “Convenient Synthesis of 2-Thioimidazolone/Menadione Conjugates via a Two-Step Sequence Starting with Direct Amination of Menadione.” SynOpen, vol. 04, no. 02, Apr. 2020, pp. 38-43. http://www.thieme-connect.de/DOI/DOI?10.1055/s-0040-1707519.