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,  том 329 ,  издание 5996 ,  страницы 1175-1180

Spiroindolones, a Potent Compound Class for the Treatment of Malaria

Тип публикации: Journal Article
Дата публикации: 2010-09-03
SCImago Q1
Tоп 10% SCImago
WOS Q1
БС1
SJR: 10.948
CiteScore: 44.6
Impact factor: 47.3
ISSN: 00368075, 10959203
Multidisciplinary
Краткое описание
Antimalarial Drug Candidate

Spiroindolones were discovered as promising antimalarial drug candidates through a high-throughput screening approach that should be applicable to a range of neglected infectious diseases. Rottmann et al. (p. 1175 ; see the Perspective by Wells ) present the preclinical profile for an optimized spiroindolone drug candidate, NITD609. They obtained evidence for a decrease in drug sensitivity in strains of the malaria parasite Plasmodium falciparum bearing amino acid mutations in the P-type ATPase, indicating possible mechanisms of action and/or resistance.

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ГОСТ |
Цитировать
Rottmann M. et al. Spiroindolones, a Potent Compound Class for the Treatment of Malaria // Science. 2010. Vol. 329. No. 5996. pp. 1175-1180.
ГОСТ со всеми авторами (до 50) Скопировать
Rottmann M., McNamara C., Yeung B. K. S., Lee M. C., ZOU B., Russell B., Seitz P., Plouffe D. M., Dharia N. V., Tan J., Cohen S. B., Spencer K. R., González Páez G. E., Lakshminarayana S. B., Goh A., Suwanarusk R., Jegla T., Schmitt E. K., Beck H. P., Brun R., Nosten F., Rénia L., Dartois V., Keller T. H., Fidock D. A., Winzeler E. A., Diagana T. T. Spiroindolones, a Potent Compound Class for the Treatment of Malaria // Science. 2010. Vol. 329. No. 5996. pp. 1175-1180.
RIS |
Цитировать
TY - JOUR
DO - 10.1126/science.1193225
UR - https://doi.org/10.1126/science.1193225
TI - Spiroindolones, a Potent Compound Class for the Treatment of Malaria
T2 - Science
AU - Rottmann, Matthias
AU - McNamara, Case
AU - Yeung, Bryan K S
AU - Lee, Marcus C.S.
AU - ZOU, BIN
AU - Russell, Bruce
AU - Seitz, Patrick
AU - Plouffe, David M.
AU - Dharia, Neekesh V
AU - Tan, Jocelyn
AU - Cohen, Steven B.
AU - Spencer, Kathryn R
AU - González Páez, Gonzalo E
AU - Lakshminarayana, Suresh B
AU - Goh, Anne
AU - Suwanarusk, Rossarin
AU - Jegla, Timothy
AU - Schmitt, Esther K.
AU - Beck, Hans Peter
AU - Brun, Reto
AU - Nosten, François
AU - Rénia, Laurent
AU - Dartois, Véronique
AU - Keller, Thomas H.
AU - Fidock, David A.
AU - Winzeler, Elizabeth A
AU - Diagana, Thierry T
PY - 2010
DA - 2010/09/03
PB - American Association for the Advancement of Science (AAAS)
SP - 1175-1180
IS - 5996
VL - 329
PMID - 20813948
SN - 0036-8075
SN - 1095-9203
ER -
BibTex |
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BibTex (до 50 авторов) Скопировать
@article{2010_Rottmann,
author = {Matthias Rottmann and Case McNamara and Bryan K S Yeung and Marcus C.S. Lee and BIN ZOU and Bruce Russell and Patrick Seitz and David M. Plouffe and Neekesh V Dharia and Jocelyn Tan and Steven B. Cohen and Kathryn R Spencer and Gonzalo E González Páez and Suresh B Lakshminarayana and Anne Goh and Rossarin Suwanarusk and Timothy Jegla and Esther K. Schmitt and Hans Peter Beck and Reto Brun and François Nosten and Laurent Rénia and Véronique Dartois and Thomas H. Keller and David A. Fidock and Elizabeth A Winzeler and Thierry T Diagana},
title = {Spiroindolones, a Potent Compound Class for the Treatment of Malaria},
journal = {Science},
year = {2010},
volume = {329},
publisher = {American Association for the Advancement of Science (AAAS)},
month = {sep},
url = {https://doi.org/10.1126/science.1193225},
number = {5996},
pages = {1175--1180},
doi = {10.1126/science.1193225}
}
MLA
Цитировать
Rottmann, Matthias, et al. “Spiroindolones, a Potent Compound Class for the Treatment of Malaria.” Science, vol. 329, no. 5996, Sep. 2010, pp. 1175-1180. https://doi.org/10.1126/science.1193225.
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