The neuroleptic activity of haloperidol increases after its solubilization in surfactant micelles
Тип публикации: Journal Article
Дата публикации: 1989-12-04
SCImago Q1
Tоп 10% SCImago
WOS Q2
БС1
SJR: 1.181
CiteScore: 6.1
Impact factor: 3
ISSN: 00145793, 18733468
PubMed ID:
2599097
Biochemistry
Molecular Biology
Cell Biology
Genetics
Structural Biology
Biophysics
Краткое описание
It has been suggested to use surfactant micelles as microcontainers for increasing the efficiency of neuroleptic targeting from blood flow into the brain. The neuroleptic action of haloperidol, intraperitoneally injected into mice in micellar solution of non‐ionic block copolymer surfactant (pluronic P‐85) in water, increased several‐fold if compared with that observed for haloperidol aqueous solution. Incorporation of brain‐specific antibodies into haloperidol‐containing micelles resulted in additional drastic increase (more than by 2 orders of magnitude) in the drug effect.
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KABANOV A. et al. The neuroleptic activity of haloperidol increases after its solubilization in surfactant micelles // FEBS Letters. 1989. Vol. 258. No. 2. pp. 343-345.
ГОСТ со всеми авторами (до 50)
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KABANOV A., Chekhonin V. P., Alakhov V. Yu., Batrakova E. V., Lebedev A. S., Melik-Nubarov N., Arzhakov S. A., Levashov A. V., Morozov G. V., Severin E. S., Kabanov V. The neuroleptic activity of haloperidol increases after its solubilization in surfactant micelles // FEBS Letters. 1989. Vol. 258. No. 2. pp. 343-345.
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TY - JOUR
DO - 10.1016/0014-5793(89)81689-8
UR - https://febs.onlinelibrary.wiley.com/doi/10.1016/0014-5793(89)81689-8
TI - The neuroleptic activity of haloperidol increases after its solubilization in surfactant micelles
T2 - FEBS Letters
AU - KABANOV, A.V.
AU - Chekhonin, V. P.
AU - Alakhov, V Yu
AU - Batrakova, E V
AU - Lebedev, A. S.
AU - Melik-Nubarov, N.S.
AU - Arzhakov, S A
AU - Levashov, A V
AU - Morozov, G V
AU - Severin, E S.
AU - Kabanov, V.A.
PY - 1989
DA - 1989/12/04
PB - Wiley
SP - 343-345
IS - 2
VL - 258
PMID - 2599097
SN - 0014-5793
SN - 1873-3468
ER -
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BibTex (до 50 авторов)
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@article{1989_KABANOV,
author = {A.V. KABANOV and V. P. Chekhonin and V Yu Alakhov and E V Batrakova and A. S. Lebedev and N.S. Melik-Nubarov and S A Arzhakov and A V Levashov and G V Morozov and E S. Severin and V.A. Kabanov},
title = {The neuroleptic activity of haloperidol increases after its solubilization in surfactant micelles},
journal = {FEBS Letters},
year = {1989},
volume = {258},
publisher = {Wiley},
month = {dec},
url = {https://febs.onlinelibrary.wiley.com/doi/10.1016/0014-5793(89)81689-8},
number = {2},
pages = {343--345},
doi = {10.1016/0014-5793(89)81689-8}
}
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MLA
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KABANOV, A.V., et al. “The neuroleptic activity of haloperidol increases after its solubilization in surfactant micelles.” FEBS Letters, vol. 258, no. 2, Dec. 1989, pp. 343-345. https://febs.onlinelibrary.wiley.com/doi/10.1016/0014-5793(89)81689-8.
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