Organic and Biomolecular Chemistry, volume 18, issue 16, pages 3069-3081
Proof of concept for poor inhibitor binding and efficient formation of covalent adducts of KRASG12C and ARS compounds
Publication type: Journal Article
Publication date: 2020-02-19
Journal:
Organic and Biomolecular Chemistry
Quartile SCImago
Q1
Quartile WOS
Q2
Impact factor: 3.2
ISSN: 14770520, 14770539
Organic Chemistry
Biochemistry
Physical and Theoretical Chemistry
Abstract
Comprehensive molecular modeling and kinetic analysis reveal a novel mechanism of the inhibition of the oncogenic mutant of the “undruggable” KRAS protein.
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1 publication, 6.25%
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1 publication, 6.25%
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1 publication, 6.25%
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Citations by publishers
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1
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4
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Multidisciplinary Digital Publishing Institute (MDPI)
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4 publications, 25%
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Elsevier
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2 publications, 12.5%
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Royal Society of Chemistry (RSC)
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2 publications, 12.5%
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American Chemical Society (ACS)
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2 publications, 12.5%
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Springer Nature
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2 publications, 12.5%
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Future Medicine
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1 publication, 6.25%
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American Society for Biochemistry and Molecular Biology
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1 publication, 6.25%
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Wiley
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Wiley
1 publication, 6.25%
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4
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- We do not take into account publications that without a DOI.
- Statistics recalculated only for publications connected to researchers, organizations and labs registered on the platform.
- Statistics recalculated weekly.
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GOST
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Khrenova M. G. et al. Proof of concept for poor inhibitor binding and efficient formation of covalent adducts of KRASG12C and ARS compounds // Organic and Biomolecular Chemistry. 2020. Vol. 18. No. 16. pp. 3069-3081.
GOST all authors (up to 50)
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Khrenova M. G., Kulakova A. M., Nemukhin A. Proof of concept for poor inhibitor binding and efficient formation of covalent adducts of KRASG12C and ARS compounds // Organic and Biomolecular Chemistry. 2020. Vol. 18. No. 16. pp. 3069-3081.
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RIS
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TY - JOUR
DO - 10.1039/d0ob00071j
UR - https://doi.org/10.1039%2Fd0ob00071j
TI - Proof of concept for poor inhibitor binding and efficient formation of covalent adducts of KRASG12C and ARS compounds
T2 - Organic and Biomolecular Chemistry
AU - Khrenova, Maria G.
AU - Kulakova, Anna M
AU - Nemukhin, Alexander
PY - 2020
DA - 2020/02/19 00:00:00
PB - Royal Society of Chemistry (RSC)
SP - 3069-3081
IS - 16
VL - 18
SN - 1477-0520
SN - 1477-0539
ER -
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BibTex
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@article{2020_Khrenova,
author = {Maria G. Khrenova and Anna M Kulakova and Alexander Nemukhin},
title = {Proof of concept for poor inhibitor binding and efficient formation of covalent adducts of KRASG12C and ARS compounds},
journal = {Organic and Biomolecular Chemistry},
year = {2020},
volume = {18},
publisher = {Royal Society of Chemistry (RSC)},
month = {feb},
url = {https://doi.org/10.1039%2Fd0ob00071j},
number = {16},
pages = {3069--3081},
doi = {10.1039/d0ob00071j}
}
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MLA
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Khrenova, Maria G., et al. “Proof of concept for poor inhibitor binding and efficient formation of covalent adducts of KRASG12C and ARS compounds.” Organic and Biomolecular Chemistry, vol. 18, no. 16, Feb. 2020, pp. 3069-3081. https://doi.org/10.1039%2Fd0ob00071j.