5,7-Dimethoxyflavone induces melanogenesis in B16F10 melanoma cells through cAMP-dependent signalling
Тип публикации: Journal Article
Дата публикации: 2011-03-22
SCImago Q1
Tоп 10% SCImago
WOS Q2
БС1
SJR: 1.068
CiteScore: 6.7
Impact factor: 3.1
ISSN: 09066705, 16000625
PubMed ID:
21426409
Biochemistry
Molecular Biology
Dermatology
Краткое описание
Melanin protects the skin against ultraviolet radiation (UVR) and diverse free radicals. Agents that increase melanin synthesis in melanocytes may reduce UVR-induced skin damage and skin cancer. In the present study, we evaluated the effects of 5,7-dimethoxyflavone (5,7-DMF) on melanogenic protein expression and signalling pathways. We found that 5,7-DMF significantly increased melanin content by upregulating microphthalmia-associated transcription factor and related melanogenic proteins. Additionally, 5,7-DMF increased cAMP levels, which activates a cascade of reactions, such as cAMP responsive element-binding protein and Akt/glycogen synthase kinase-3β (GSK-3β) signalling. Thus, 5,7-DMF may be an effective pigmentation stimulator for photoprotection and hypopigmentation disorders.
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ГОСТ
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Kang Y. G. et al. 5,7-Dimethoxyflavone induces melanogenesis in B16F10 melanoma cells through cAMP-dependent signalling // Experimental Dermatology. 2011. Vol. 20. No. 5. pp. 445-447.
ГОСТ со всеми авторами (до 50)
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Kang Y. G., Choi E. J., Choi Y., Hwang J. K. 5,7-Dimethoxyflavone induces melanogenesis in B16F10 melanoma cells through cAMP-dependent signalling // Experimental Dermatology. 2011. Vol. 20. No. 5. pp. 445-447.
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TY - JOUR
DO - 10.1111/j.1600-0625.2010.01236.x
UR - https://doi.org/10.1111/j.1600-0625.2010.01236.x
TI - 5,7-Dimethoxyflavone induces melanogenesis in B16F10 melanoma cells through cAMP-dependent signalling
T2 - Experimental Dermatology
AU - Kang, Young Gyu
AU - Choi, Eun Jung
AU - Choi, Yuri
AU - Hwang, Jae Kwan
PY - 2011
DA - 2011/03/22
PB - Wiley
SP - 445-447
IS - 5
VL - 20
PMID - 21426409
SN - 0906-6705
SN - 1600-0625
ER -
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BibTex (до 50 авторов)
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@article{2011_Kang,
author = {Young Gyu Kang and Eun Jung Choi and Yuri Choi and Jae Kwan Hwang},
title = {5,7-Dimethoxyflavone induces melanogenesis in B16F10 melanoma cells through cAMP-dependent signalling},
journal = {Experimental Dermatology},
year = {2011},
volume = {20},
publisher = {Wiley},
month = {mar},
url = {https://doi.org/10.1111/j.1600-0625.2010.01236.x},
number = {5},
pages = {445--447},
doi = {10.1111/j.1600-0625.2010.01236.x}
}
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MLA
Скопировать
Kang, Young Gyu, et al. “5,7-Dimethoxyflavone induces melanogenesis in B16F10 melanoma cells through cAMP-dependent signalling.” Experimental Dermatology, vol. 20, no. 5, Mar. 2011, pp. 445-447. https://doi.org/10.1111/j.1600-0625.2010.01236.x.
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