Antitumor Activity of Fascaplysin Derivatives on Glioblastoma Model In Vitro
Тип публикации: Journal Article
Дата публикации: 2018-03-25
Включен в RSCI
scimago Q3
wos Q4
БС2
SJR: 0.277
CiteScore: 1.5
Impact factor: 0.6
ISSN: 00074888, 15738221, 03659615, 24131008
PubMed ID:
29577186
General Biochemistry, Genetics and Molecular Biology
General Medicine
Краткое описание
Antitumor efficiency of fascaplysin synthetic derivatives (7-phenylfascaplysin, 3-chlorofascaplysin, 3-bromofascaplysin, and 10-bromofascaplysin) was compared out in vitro on C6 glioma cells. The cytotoxic efficiency of all tested compounds was higher than that of unsubstituted fascaplysin; 3-bromofascaplysin and 7-phenylfascaplysin exhibited the best capacity to kill glioma C6 cells. Apoptosis was the main mechanism of glioma cell death. The cytotoxic activity of these compounds increased with prolongation of exposure to the substance and increase of its concentration. Fascaplysin derivatives modified all phases of glioma cell vital cycle. The count of viable tumor cell in G0 phase remained minimum by the end of experiment under the effects of 3-bromofascaplysin and 7-phenylfascaplysin.
Найдено
Ничего не найдено, попробуйте изменить настройки фильтра.
Найдено
Ничего не найдено, попробуйте изменить настройки фильтра.
Топ-30
Журналы
|
1
2
3
4
5
6
7
8
|
|
|
Marine Drugs
8 публикаций, 50%
|
|
|
International Review of Neurobiology
2 публикации, 12.5%
|
|
|
Biomedicines
1 публикация, 6.25%
|
|
|
Biomedicine and Pharmacotherapy
1 публикация, 6.25%
|
|
|
ChemistrySelect
1 публикация, 6.25%
|
|
|
Studies in Natural Products Chemistry
1 публикация, 6.25%
|
|
|
Molecules
1 публикация, 6.25%
|
|
|
Bioorganic and Medicinal Chemistry
1 публикация, 6.25%
|
|
|
1
2
3
4
5
6
7
8
|
Издатели
|
2
4
6
8
10
|
|
|
MDPI
10 публикаций, 62.5%
|
|
|
Elsevier
5 публикаций, 31.25%
|
|
|
Wiley
1 публикация, 6.25%
|
|
|
2
4
6
8
10
|
- Мы не учитываем публикации, у которых нет DOI.
- Статистика публикаций обновляется еженедельно.
Вы ученый?
Создайте профиль, чтобы получать персональные рекомендации коллег, конференций и новых статей.
Метрики
16
Всего цитирований:
16
Цитирований c 2025:
1
(6.25%)
Цитировать
ГОСТ |
RIS |
BibTex |
MLA
Цитировать
ГОСТ
Скопировать
Lyakhova I. A. et al. Antitumor Activity of Fascaplysin Derivatives on Glioblastoma Model In Vitro // Bulletin of Experimental Biology and Medicine. 2018. Vol. 164. No. 5. pp. 666-672.
ГОСТ со всеми авторами (до 50)
Скопировать
Lyakhova I. A., Bryukhovetsky I. S., Kudryavtsev I. V., Khotimchenko Yu. S., Zhidkov M. E., Kantemirov A. V. Antitumor Activity of Fascaplysin Derivatives on Glioblastoma Model In Vitro // Bulletin of Experimental Biology and Medicine. 2018. Vol. 164. No. 5. pp. 666-672.
Цитировать
RIS
Скопировать
TY - JOUR
DO - 10.1007/s10517-018-4055-4
UR - https://doi.org/10.1007/s10517-018-4055-4
TI - Antitumor Activity of Fascaplysin Derivatives on Glioblastoma Model In Vitro
T2 - Bulletin of Experimental Biology and Medicine
AU - Lyakhova, I A
AU - Bryukhovetsky, I S
AU - Kudryavtsev, I. V.
AU - Khotimchenko, Yu S
AU - Zhidkov, M E
AU - Kantemirov, A V
PY - 2018
DA - 2018/03/25
PB - Springer Nature
SP - 666-672
IS - 5
VL - 164
PMID - 29577186
SN - 0007-4888
SN - 1573-8221
SN - 0365-9615
SN - 2413-1008
ER -
Цитировать
BibTex (до 50 авторов)
Скопировать
@article{2018_Lyakhova,
author = {I A Lyakhova and I S Bryukhovetsky and I. V. Kudryavtsev and Yu S Khotimchenko and M E Zhidkov and A V Kantemirov},
title = {Antitumor Activity of Fascaplysin Derivatives on Glioblastoma Model In Vitro},
journal = {Bulletin of Experimental Biology and Medicine},
year = {2018},
volume = {164},
publisher = {Springer Nature},
month = {mar},
url = {https://doi.org/10.1007/s10517-018-4055-4},
number = {5},
pages = {666--672},
doi = {10.1007/s10517-018-4055-4}
}
Цитировать
MLA
Скопировать
Lyakhova, I. A., et al. “Antitumor Activity of Fascaplysin Derivatives on Glioblastoma Model In Vitro.” Bulletin of Experimental Biology and Medicine, vol. 164, no. 5, Mar. 2018, pp. 666-672. https://doi.org/10.1007/s10517-018-4055-4.
Лаборатории
Профили